SCHEMBL9499780

SCHEMBL9499780

COc1ccc(N2CCC(C=O)CC2)cc1OC

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.52
DPP4 P27487 7/20 0.48
CYP1A2 P05177 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
HIF1A Q16665 3/20 0.44
MAOB P27338 1/20 0.44
LMNA P02545 2/20 0.43
MAPT P10636 1/20 0.43
CTSB P07858 1/20 0.43
CTSS P25774 1/20 0.43
CTSK P43235 1/20 0.43
NPC1 O15118 1/20 0.43
POLB P06746 1/20 0.43
RAB9A P51151 1/20 0.43
HTR7 P34969 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9503509 0.98 ALDH1A1 (0.51) ALDH1A1DPP4CYP1A2L3MBTL1HIF1A
Hydrochloric Acid SCHEMBL17870560 0.87 ALDH1A1 (0.46) ALDH1A1DPP4MAOBLMNAMAPT
Hydrochloric Acid SCHEMBL17870558 0.86 ALDH1A1 (0.45) ALDH1A1MAOBLMNAMAPT
SCHEMBL31458389 0.83 ALDH1A1 (0.70) ALDH1A1CYP1A2L3MBTL1LMNAMAPT
SCHEMBL28859927 0.83 ALDH1A1 (0.70) ALDH1A1CYP1A2L3MBTL1LMNAMAPT
SCHEMBL230404 0.80 HTR3E (0.53) ALDH1A1L3MBTL1LMNAMAPTPOLB
SCHEMBL9499769 0.79 CTSB (0.51) ALDH1A1DPP4HIF1ACTSBCTSS
SCHEMBL12716971 0.78 NEK2 (0.54) DPP4HIF1ACTSBCTSSCTSK
Hydrochloric Acid SCHEMBL9503502 0.78 CTSB (0.50) ALDH1A1DPP4HIF1ACTSBCTSS
SCHEMBL24833007 0.77 ALDH1A1 (0.40) ALDH1A1L3MBTL1MAOBLMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0325268-B1 1,4-DISUBSTITUTED-PIPERIDINYL COMPOUNDS MERRELL DOW PHARMACEUTICALS INC. (US) 1993-06-02 EP disclosed
US-5162342-A USE OF 1,4-DISUBSTITUTED-PIPERIDINYL COMPOUNDS FOR ANALGESIA AND MUSCLE RELAXATION MERRELL DOW PHARMACEUTICALS INC. (US) 1992-11-10 US disclosed
US-5064838-A 1,4-DISUBSTITUTED-PIPERIDINYL COMPOUNDS AS PAIN RELIEVERS MERRELL DOW PHARMACEUTICALS (US) 1991-11-12 US disclosed
CN-1035823-A 1, the 4-Disubstituted-piperidnyl compounds MERRELL DOW PHARMA (US) 1989-09-27 CN disclosed
EP-0325268-A1 1,4-Disubstituted-piperidinyl compounds MERRELL DOW PHARMACEUTICALS INC. (US) 1989-07-26 EP disclosed