SCHEMBL9501323

SCHEMBL9501323

c1ccc2c(c1)CCN2Cc1ccncc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.58
ALOX15 P16050 2/20 0.58
MEN1 O00255 2/20 0.58
KMT2A Q03164 2/20 0.58
USP2 O75604 1/20 0.58
CDK4 P11802 1/20 0.58
CCND1 P24385 1/20 0.58
TAAR1 Q96RJ0 2/20 0.56
TRPM5 Q9NZQ8 1/20 0.52
TRPV1 Q8NER1 3/20 0.49
GAA P10253 2/20 0.48
KDM4E B2RXH2 2/20 0.47
MAPT P10636 2/20 0.47
LMNA P02545 1/20 0.47
PTK2B Q14289 1/20 0.47
ESR2 Q92731 1/20 0.47
TSHR P16473 1/20 0.47
HDAC1 Q13547 2/20 0.47
HDAC6 Q9UBN7 2/20 0.47
HDAC3 O15379 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29875634 0.86 ALDH1A1 (0.66) ALDH1A1ALOX15MEN1KMT2AUSP2
SCHEMBL29558 0.86 ALDH1A1 (0.66) ALDH1A1ALOX15MEN1KMT2AUSP2
SCHEMBL29351443 0.84 ALDH1A1 (0.64) ALDH1A1ALOX15MEN1KMT2AUSP2
SCHEMBL28567500 0.81 DRD4 (0.61) ALDH1A1ALOX15MEN1KMT2AUSP2
SCHEMBL3850387 0.80 ALDH1A1 (0.58) ALDH1A1ALOX15MEN1KMT2AUSP2
SCHEMBL3096260 0.80 ALDH1A1 (0.58) ALDH1A1ALOX15MEN1KMT2AUSP2
SCHEMBL3098204 0.80 ALDH1A1 (0.58) ALDH1A1ALOX15MEN1KMT2AUSP2
SCHEMBL15447287 0.80 ALDH1A1 (0.58) ALDH1A1ALOX15MEN1KMT2AUSP2
SCHEMBL29571652 0.80 ALDH1A1 (0.58) ALDH1A1ALOX15MEN1KMT2AUSP2
SCHEMBL25185012 0.80 TRPM5 (0.59) ALDH1A1ALOX15MEN1KMT2AUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5214058-A Acetylcholinesterase inhibitors, treatment of senile dementia HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1993-05-25 US disclosed
EP-0471296-A1 1-(Pyridinylalkyl)-1H-indoles, indolines and related analogs HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-02-19 EP disclosed