SCHEMBL9501563

SCHEMBL9501563

O=S(=O)(Nc1ccccc1OC1CCCCC1)C(F)(F)F

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MRGPRX1 Q96LB2 1/20 0.49
PTGS2 P35354 10/20 0.48
PTGS1 P23219 9/20 0.48
CA2 P00918 1/20 0.46
CYP19A1 P11511 2/20 0.43
ALDH1A1 P00352 2/20 0.43
MEN1 O00255 1/20 0.43
PTGES O14684 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
MAPT P10636 1/20 0.43
ALOX15 P16050 1/20 0.43
TSHR P16473 1/20 0.43
CYP2C19 P33261 1/20 0.43
KMT2A Q03164 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
SLC22A12 Q96S37 2/20 0.41
PDE4D Q08499 2/20 0.40
FABP4 P15090 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8523784 0.81 PTGS1 (0.61) MRGPRX1PTGS2PTGS1CYP19A1ALDH1A1
SCHEMBL9501964 0.78 CYP19A1 (0.73) PTGS2PTGS1CYP19A1ALDH1A1MEN1
SCHEMBL9502671 0.77 CYP19A1 (0.72) PTGS2PTGS1CYP19A1ALDH1A1MEN1
SCHEMBL9502677 0.77 CYP19A1 (0.72) PTGS2PTGS1CYP19A1ALDH1A1MEN1
SCHEMBL9502689 0.77 CYP19A1 (0.72) PTGS2PTGS1CYP19A1ALDH1A1MEN1
SCHEMBL9502681 0.77 CYP19A1 (0.56) MRGPRX1PTGS2PTGS1CA2CYP19A1
SCHEMBL27595683 0.77 PTGS1 (0.59) PTGS2PTGS1CA2SLC22A12
SCHEMBL9502643 0.76 CYP19A1 (0.73) PTGS2PTGS1CYP19A1ALDH1A1MEN1
SCHEMBL28754288 0.75 TSHR (0.50) MRGPRX1PTGS2MAPTTSHRSMN1; SMN2
SCHEMBL649744 0.72 PTGS1 (0.70) PTGS2PTGS1CA2TSHRSLC22A12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0317332-B1 SULFONANILIDE COMPOUNDS TAISHO PHARMACEUTICAL CO. LTD (JP) 1993-05-19 EP disclosed
US-4885367-A ANTIINFLAMMATORY AGENTS, ANTIPYRETICS, ANALGESICS; SIDE EFFECT REDUCTION TAISHO PHARMACEUTICAL CO., LTD. (JP) 1989-12-05 US disclosed
EP-0317332-A2 Sulfonanilide compounds TAISHO PHARMACEUTICAL CO. LTD (JP) 1989-05-24 EP disclosed