SCHEMBL9501924

SCHEMBL9501924

Cc1ccnc(-c2cccc(C(C)c3ccccc3)n2)n1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 1/20 0.38
GRM5 P41594 3/20 0.36
TGFBR1 P36897 4/20 0.35
CCR1 P32246 1/20 0.34
CCR8 P51685 1/20 0.34
COMT P21964 3/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33
HTT P42858 1/20 0.33
RECQL P46063 1/20 0.33
PIM1 P11309 1/20 0.33
PIM2 Q9P1W9 1/20 0.33
IDH1 O75874 1/20 0.33
KDM4A O75164 1/20 0.32
KDM4C Q9H3R0 1/20 0.32
KDM5B Q9UGL1 1/20 0.32
MAPK14 Q16539 1/20 0.32
TSHR P16473 1/20 0.32
POLB P06746 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9586361 0.88 GRM5 (0.42) IRAK4GRM5TGFBR1CCR1CCR8
SCHEMBL4333513 0.78 HTT (0.50) GRM5CCR1CCR8SLC6A2SLC6A4
SCHEMBL15470589 0.76 CCR1 (0.60) GRM5TGFBR1CCR1CCR8IDH1
SCHEMBL8854902 0.75 MEN1 (0.55) GRM5TGFBR1CCR1CCR8
SCHEMBL6559740 0.74 KMT2A (0.41) SLC6A2SLC6A4SLC6A3PIM1PIM2
SCHEMBL9500899 0.72 BRD4 (0.41) GRM5TGFBR1CCR1CCR8POLB
SCHEMBL7964553 0.71 KDM4E (0.59) GRM5CCR1CCR8HTTPOLB
SCHEMBL9026653 0.70 CCR1 (0.42) GRM5TGFBR1CCR1CCR8MAPK14
SCHEMBL10539132 0.69 CYP2A6 (0.53) GRM5TGFBR1CCR1CCR8MAPK14
SCHEMBL9031119 0.69 GRM4 (0.62) GRM5TSHRPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5185339-A FUNGICIDAL COMPOUNDS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-02-09 US disclosed
EP-0459662-A1 Fungicidal compounds ZENECA LIMITED (GB) 1991-12-04 EP disclosed