SCHEMBL9502395

SCHEMBL9502395

CCOC(=O)C1=C(CCl)NC(C(OCC)OCC)=C(C(=O)OCC)C1c1cccc(Cl)c1

nearest known ligand 0.49

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 7/20 0.46
CACNA1F O60840 2/20 0.46
CACNA1D Q01668 2/20 0.46
CACNA1S Q13698 2/20 0.46
CACNA1C Q13936 2/20 0.46
ABCC1 P33527 1/20 0.44
ADORA3 P0DMS8 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9518607 0.85 CACNA1B (0.41) CACNA1BCACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL9513394 0.85 ABCC1 (0.58) CACNA1BCACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL9504268 0.84 CACNA1F (0.50) CACNA1BCACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL9519468 0.80 CACNA1F (0.47) CACNA1BCACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL3026966 0.78 ABCC1 (0.71) CACNA1BCACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL7380442 0.77 KIF11 (0.56) CACNA1FCACNA1DCACNA1SCACNA1CABCC1
SCHEMBL11773488 0.77 CACNA1F (0.56) CACNA1BCACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL11522715 0.76 ABCC1 (0.58) CACNA1BCACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL9675983 0.75 ABCC1 (0.57) CACNA1BCACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL11459111 0.74 ABCC1 (0.55) CACNA1BCACNA1FCACNA1DCACNA1SCACNA1C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0458823-B1 A PROCESS FOR PREPARATION OF ENANTIOMERICALLY PURE POLYSUBSTITUTED 1,4-DIHYDROPYRIDINES BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1993-10-13 EP disclosed
US-5245039-A PROCESS FOR PREPARATION OF ENANTIOMERICALLY PURE POLYSUBSTITUTED 1,4-DIHYDROPYRIDINES BOEHRINGER MANNHEIM ITALIA (IT) 1993-09-14 US disclosed
EP-0458823-A1 A PROCESS FOR PREPARATION OF ENANTIOMERICALLY PURE POLYSUBSTITUTED 1,4-DIHYDROPYRIDINES. BOEHRINGER MANNHEIM ITALIA (IT) 1991-12-04 EP disclosed
WO-1990009376-A1 A PROCESS FOR PREPARATION OF ENANTIOMERICALLY PURE POLYSUBSTITUTED 1,4-DIHYDROPYRIDINES BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1990-08-23 WO disclosed
EP-0383320-A1 A process for preparation of enantiomerically pure polysubstituted 1,4-dihydropyridines BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1990-08-22 EP disclosed