SCHEMBL9502744

SCHEMBL9502744

Cc1cccc2nc(C(F)(F)F)[nH]c12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 3/20 0.53
PKM P14618 1/20 0.47
MAPT P10636 5/20 0.44
HPGD P15428 4/20 0.44
KDM4E B2RXH2 4/20 0.44
POLB P06746 2/20 0.44
AR P10275 1/20 0.42
ELANE P08246 1/20 0.40
ALDH1A1 P00352 3/20 0.39
GAA P10253 2/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
ALOX15 P16050 1/20 0.39
CYP2C19 P33261 1/20 0.39
HSD17B10 Q99714 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
PARP1 P09874 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5508549 0.84 MEN1 (0.40) NPSR1HPGDARELANEALDH1A1
SCHEMBL6759198 0.84 ADORA3 (0.40) NPSR1HPGDARALDH1A1L3MBTL1
SCHEMBL1128774 0.81 NPSR1 (0.37) NPSR1HPGDARALDH1A1MEN1
SCHEMBL28344139 0.80 NPSR1 (0.55) NPSR1PKMMAPTHPGDKDM4E
SCHEMBL11835605 0.79 NPSR1 (0.50) NPSR1PKMMAPTHPGDKDM4E
SCHEMBL9504950 0.79 NPSR1 (0.53) NPSR1PKMMAPTHPGDKDM4E
SCHEMBL1663646 0.79 MAPT (0.54) NPSR1PKMMAPTHPGDKDM4E
SCHEMBL12145773 0.78 NPSR1 (0.55) NPSR1PKMMAPTHPGDKDM4E
SCHEMBL6957142 0.78 NPSR1 (0.49) NPSR1PKMHPGDKDM4EELANE
SCHEMBL10722861 0.76 NPSR1 (0.50) NPSR1PKMMAPTHPGDKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117534620-A Preparation method of palladium-catalyzed hydrocarbon bond functionalized 2-trifluoromethyl benzimidazole compound 六盘水师范学院 2024-02-09 CN disclosed
EP-0186190-B1 BENZIMIDAZOLE DERIVATIVES, AND THEIR PRODUCTION AND USE SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1993-05-26 EP disclosed
US-4663339-A Acaricidal and insecticidal substituted 1-phenylalkylbenzimidazoles SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1987-05-05 US disclosed
EP-0186190-A2 Benzimidazole derivatives, and their production and use SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1986-07-02 EP disclosed