SCHEMBL9502893

SCHEMBL9502893

Nc1nc(Cl)c2ncn(Cc3cccc(OCP(=O)(O)O)c3)c2n1

nearest known ligand 0.69

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PNP P00491 6/20 0.69
HDAC6 Q9UBN7 7/20 0.54
HDAC1 Q13547 5/20 0.54
HDAC4 P56524 1/20 0.54
HSP90AA1 P07900 3/20 0.52
HSP90AB1 P08238 3/20 0.52
HDAC2 Q92769 1/20 0.52
ADORA2A P29274 2/20 0.49
ADORA1 P30542 2/20 0.49
YTHDC1 Q96MU7 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9504559 0.88 HDAC6 (0.62) PNPHDAC6HDAC1HDAC4HSP90AA1
SCHEMBL9506694 0.87 PNP (0.70) PNPHDAC6HDAC1HDAC4HSP90AA1
SCHEMBL3394076 0.84 HSP90AB1 (0.68) HDAC6HDAC1HDAC4HSP90AA1HSP90AB1
SCHEMBL9506062 0.82 PNP (1.00) PNP
SCHEMBL3394097 0.81 HDAC6 (0.60) PNPHDAC6HDAC1HDAC4HSP90AA1
SCHEMBL9504540 0.81 PNP (0.69) PNPHDAC6HDAC1HDAC4HSP90AA1
SCHEMBL9504737 0.79 PNP (0.68) PNPHDAC6HDAC1HDAC4HSP90AA1
SCHEMBL6272417 0.78 ALDH1A1 (0.66) PNPHDAC6HDAC1HDAC4HSP90AA1
SCHEMBL9502871 0.77 HSP90AA1 (0.53) HDAC6HDAC1HDAC4HSP90AA1HSP90AB1
SCHEMBL5469402 0.76 HDAC6 (0.61) HDAC6HDAC1HDAC4HSP90AA1HSP90AB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0550574-A1 HETEROCYCLIC COMPOUNDS THE WELLCOME FOUNDATION LIMITED (GB) 1993-07-14 EP disclosed
WO-1992005180-A1 HETEROCYCLIC COMPOUNDS THE WELLCOME FOUNDATION LIMITED (GB) 1992-04-02 WO disclosed