SCHEMBL9503225

SCHEMBL9503225

CNc1c(-c2nncs2)cc(C(C)(C)C)c(O)c1C(C)(C)C

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 15/20 0.43
PTGS2 P35354 11/20 0.43
GAA P10253 1/20 0.32
CA2 P00918 2/20 0.32
CA1 P00915 1/20 0.32
GLRA3 O75311 1/20 0.31
GLRB P48167 1/20 0.31
ALDH1A1 P00352 1/20 0.31
POLB P06746 1/20 0.31
TYR P14679 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
ALOX5 P09917 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8766812 0.71 PTGS1 (0.58) PTGS1PTGS2CA2CA1ALOX5
SCHEMBL8152293 0.70 CYP2C19 (0.46) PTGS1PTGS2GAACA2CA1
SCHEMBL15173818 0.66 CA2 (0.59) PTGS1PTGS2GAACA2CA1
SCHEMBL515839 0.61 ALDH1A1 (0.56) PTGS1PTGS2GAACA2CA1
SCHEMBL9180823 0.60 PTGS1 (1.00) PTGS1PTGS2CA2CA1ALOX5
SCHEMBL13400274 0.60 SMN1; SMN2 (0.54) PTGS1PTGS2GAACA2CA1
SCHEMBL27943614 0.59 CA2 (0.61) PTGS1PTGS2GAACA2CA1
SCHEMBL9731608 0.59 HPN (0.49) PTGS1PTGS2CA2CA1ALDH1A1
SCHEMBL11521507 0.58 CA2 (0.48) PTGS1PTGS2GAACA2CA1
SCHEMBL20657093 0.57 CA2 (0.65) GAACA2CA1GLRA3GLRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5256680-A 3,5-di-tertiary-butyl-4-hydroxyphenyl-1,3,4-thiadiazoles, and oxadiazoles and 3,5-di-tertiary-butyl-4-hydroxy-phenyl-1,2,4-thiadazoles, oxadiazoles and triazoles as antiinflammatory agents WARNER-LAMBERT COMPANY (US) 1993-10-26 US disclosed