SCHEMBL9503395

SCHEMBL9503395

OCCCc1cc(Br)ccc1Cl

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.42
SMN1; SMN2 Q16637 2/20 0.39
NPSR1 Q6W5P4 2/20 0.39
LMNA P02545 1/20 0.39
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
MCL1 Q07820 2/20 0.35
MAPK1 P28482 1/20 0.35
HTR2A P28223 1/20 0.35
SLC6A4 P31645 1/20 0.35
KCNH2 Q12809 1/20 0.35
STAT3 P40763 1/20 0.35
TRPV1 Q8NER1 1/20 0.34
HPGD P15428 1/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.33
PNMT P11086 1/20 0.33
TLR8 Q9NR97 1/20 0.33
CYP1A2 P05177 1/20 0.33
CA2 P00918 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3455233 0.88 SMN1; SMN2 (0.40) ALDH1A1SMN1; SMN2NPSR1LMNAMAPK1
SCHEMBL499730 0.83 CYP11B1 (0.38) ALDH1A1SMN1; SMN2NPSR1LMNACYP11B1
SCHEMBL81974 0.80 IDO1 (0.42) ALDH1A1SMN1; SMN2LMNAHPGDTLR8
SCHEMBL154181 0.79 PTGDR2 (0.44) ALDH1A1SMN1; SMN2NPSR1LMNAMAPK1
SCHEMBL6681997 0.79 ABL1 (0.41) ALDH1A1SMN1; SMN2NPSR1LMNAHTR2A
SCHEMBL2122564 0.78 TSHR (0.46) ALDH1A1SMN1; SMN2LMNAMCL1HPGD
SCHEMBL1487566 0.77 CA2 (0.42) SMN1; SMN2CYP11B1CYP11B2MCL1PTGDR2
SCHEMBL16955926 0.77 CA2 (0.39) ALDH1A1CYP11B1CYP11B2MAPK1HTR2A
SCHEMBL17399935 0.77 HPGD (0.47) ALDH1A1SMN1; SMN2LMNAHTR2ASLC6A4
SCHEMBL3455585 0.76 HTR2A (0.36) ALDH1A1SMN1; SMN2NPSR1LMNAHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993008166-A1 BENZO-ISOQUINOLINE DERIVATIVES AND ANALOGS AND THEIR USE IN THERAPEUTICS THE UPJOHN COMPANY (US) 1993-04-29 WO disclosed
EP-0539209-A1 Benzo-isoquinoline derivatives and analogs and their use in therapeutics THE UPJOHN COMPANY (US) 1993-04-28 EP disclosed