SCHEMBL9503659

SCHEMBL9503659

CC(C)CCOC(=O)Cc1ccccn1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.58
PGR P06401 1/20 0.46
ADORA3 P0DMS8 1/20 0.46
PTGS1 P23219 1/20 0.46
SLC6A2 P23975 1/20 0.46
ALDH1A1 P00352 3/20 0.46
CYP1A2 P05177 3/20 0.43
TSHR P16473 1/20 0.43
RAB9A P51151 3/20 0.42
NPC1 O15118 2/20 0.42
PTPRA P18433 1/20 0.42
HTT P42858 1/20 0.41
PPARG P37231 2/20 0.41
PPARA Q07869 1/20 0.41
MAPK1 P28482 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
LMNA P02545 1/20 0.40
HPGD P15428 1/20 0.40
HSD17B10 Q99714 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3919109 0.84 CYP19A1 (0.42) CYP19A1PGRADORA3PTGS1SLC6A2
SCHEMBL10575663 0.83 HPGD (0.49) ALDH1A1CYP1A2TSHRRAB9ANPC1
SCHEMBL3914952 0.82 CYP19A1 (0.40) CYP19A1PGRADORA3PTGS1SLC6A2
SCHEMBL356002 0.81 HSD17B10 (0.56) CYP19A1ALDH1A1CYP1A2TSHRRAB9A
SCHEMBL30858931 0.80 LMNA (0.56) ALDH1A1CYP1A2TSHRRAB9ANPC1
SCHEMBL134991 0.80 LMNA (0.56) ALDH1A1CYP1A2TSHRRAB9ANPC1
Water SCHEMBL8818123 0.79 HSD17B10 (0.55) CYP19A1ALDH1A1CYP1A2TSHRRAB9A
SCHEMBL355182 0.78 TSHR (0.57) PGRADORA3PTGS1SLC6A2ALDH1A1
SCHEMBL3916987 0.78 KMT2A (0.45) ALDH1A1CYP1A2TSHRRAB9ANPC1
SCHEMBL10573667 0.78 HSD17B10 (0.47) ALDH1A1CYP1A2TSHRRAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0336561-B1 2-PYRIDYLACETIC ACID DERIVATIVES, PREPARATIONS THEREOF, AND COMPOSITIONS CONTAINING THEM SUNTORY LIMITED (JP) 1993-07-28 EP disclosed
US-4877795-A 4H-quinolizin-4-one compounds useful for the treatment of allergic bronchial asthma, allergic rhinitis atropic dermatitis and the like KISSEI PHARMACEUTICAL CO., LTD. (JP) 1989-10-31 US disclosed
EP-0336561-A1 2-Pyridylacetic acid derivatives, preparations thereof, and compositions containing them SUNTORY LIMITED (JP) 1989-10-11 EP disclosed
US-4843083-A 2-pyridylacetic acid derivative, and pharmaceutical composition containing the same and method of treating a peptic ulcer SUNTORY LIMITED (JP) 1989-06-27 US disclosed
EP-0277755-A1 4H-quinolizin-4-one compounds exhibiting therapeutic activities Kissei Pharmaceutical Co. Ltd. (JP) 1988-08-10 EP disclosed