SCHEMBL9505256

SCHEMBL9505256

CC1=C(C(=O)O)C(c2ccccc2)C(C(=O)OCC=CC(C)(C)C)=C(C)N1

nearest known ligand 0.75

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 19/20 0.75
ADORA3 P0DMS8 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5854929 0.86 CACNA1B (1.00) CACNA1B
SCHEMBL5854934 0.86 CACNA1B (1.00) CACNA1B
SCHEMBL10475396 0.85 CACNA1B (0.74) CACNA1BADORA3
SCHEMBL10475395 0.81 ALDH1A1 (0.78) CACNA1BADORA3
SCHEMBL29173863 0.81 ADORA3 (0.82) CACNA1BADORA3
SCHEMBL5856485 0.81 CACNA1B (0.89) CACNA1B
SCHEMBL5856492 0.81 CACNA1B (0.89) CACNA1B
SCHEMBL9505249 0.79 ALDH1A1 (0.67) CACNA1BADORA3
SCHEMBL5855595 0.79 CACNA1B (0.85) CACNA1B
SCHEMBL5856555 0.79 CACNA1B (0.85) CACNA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0458823-B1 A PROCESS FOR PREPARATION OF ENANTIOMERICALLY PURE POLYSUBSTITUTED 1,4-DIHYDROPYRIDINES BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1993-10-13 EP disclosed
US-5245039-A PROCESS FOR PREPARATION OF ENANTIOMERICALLY PURE POLYSUBSTITUTED 1,4-DIHYDROPYRIDINES BOEHRINGER MANNHEIM ITALIA (IT) 1993-09-14 US disclosed
EP-0383320-A1 A process for preparation of enantiomerically pure polysubstituted 1,4-dihydropyridines BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1990-08-22 EP disclosed