SCHEMBL9505359

SCHEMBL9505359

CC1=C(C(=O)O)C(c2ccccc2)C(C(=O)O)=C(C)N1C(C)(C)C

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.49
GAA P10253 1/20 0.49
PYGM P11217 2/20 0.43
PYGL P06737 1/20 0.43
SIRT3 Q9NTG7 3/20 0.40
POLB P06746 1/20 0.40
ADORA3 P0DMS8 1/20 0.39
RIPK1 Q13546 8/20 0.38
CACNA1B Q00975 1/20 0.37
HRH3 Q9Y5N1 1/20 0.36
LMNA P02545 1/20 0.35
MEN1 O00255 1/20 0.35
MAPT P10636 1/20 0.35
HPGD P15428 1/20 0.35
TSHR P16473 1/20 0.35
HTT P42858 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16178523 0.80 KDM4E (0.66) KDM4EGAAPYGMPYGLPOLB
SCHEMBL8511172 0.74 CYP2C9 (0.45) KDM4EGAAPYGMPYGLADORA3
SCHEMBL9836397 0.73 NOTUM (0.45) KDM4EGAAPYGMPYGLPOLB
SCHEMBL9033367 0.72 PYGM (0.52) KDM4EGAAPYGMPYGLSIRT3
SCHEMBL5461012 0.72 NR3C2 (0.42) KDM4EGAAPYGMPYGLADORA3
SCHEMBL7410687 0.71 CACNA1B (0.61) GAAPOLBADORA3CACNA1BMEN1
SCHEMBL11008635 0.70 KDM4E (0.54) KDM4EGAAPYGMPYGLPOLB
SCHEMBL10445960 0.70 KDM4E (0.43) KDM4EGAAPYGMPYGLSIRT3
SCHEMBL9837158 0.69 PYGM (0.46) KDM4EGAAPYGMPYGLSIRT3
SCHEMBL16178581 0.68 TSHR (0.53) KDM4EGAALMNAMEN1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0458823-B1 A PROCESS FOR PREPARATION OF ENANTIOMERICALLY PURE POLYSUBSTITUTED 1,4-DIHYDROPYRIDINES BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1993-10-13 EP disclosed
US-5245039-A PROCESS FOR PREPARATION OF ENANTIOMERICALLY PURE POLYSUBSTITUTED 1,4-DIHYDROPYRIDINES BOEHRINGER MANNHEIM ITALIA (IT) 1993-09-14 US disclosed
EP-0458823-A1 A PROCESS FOR PREPARATION OF ENANTIOMERICALLY PURE POLYSUBSTITUTED 1,4-DIHYDROPYRIDINES. BOEHRINGER MANNHEIM ITALIA (IT) 1991-12-04 EP disclosed
WO-1990009376-A1 A PROCESS FOR PREPARATION OF ENANTIOMERICALLY PURE POLYSUBSTITUTED 1,4-DIHYDROPYRIDINES BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1990-08-23 WO disclosed
EP-0383320-A1 A process for preparation of enantiomerically pure polysubstituted 1,4-dihydropyridines BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1990-08-22 EP disclosed