SCHEMBL9836397

SCHEMBL9836397

CC1=C(C(=O)O)C(c2ccccc2)C(C(=O)O)=C(C)N1c1ccccc1C

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.45
POLB P06746 1/20 0.45
GAA P10253 2/20 0.43
MGLL Q99685 1/20 0.43
KDM4E B2RXH2 1/20 0.43
PYGM P11217 2/20 0.41
PYGL P06737 1/20 0.41
AR P10275 2/20 0.41
MAPT P10636 2/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
ALDH1A1 P00352 3/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
ELANE P08246 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
TSHR P16473 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9837076 0.85 POLB (0.64) POLBGAAKDM4EMEN1KMT2A
SCHEMBL16178523 0.78 KDM4E (0.66) POLBGAAKDM4EPYGMPYGL
SCHEMBL9505359 0.73 KDM4E (0.49) POLBGAAKDM4EPYGMPYGL
SCHEMBL9033367 0.70 PYGM (0.52) POLBGAAKDM4EPYGMPYGL
SCHEMBL7410687 0.68 CACNA1B (0.61) POLBGAAMAPTMEN1KMT2A
SCHEMBL11008635 0.68 KDM4E (0.54) POLBGAAKDM4EPYGMPYGL
SCHEMBL10445960 0.68 KDM4E (0.43) POLBGAAKDM4EPYGMPYGL
SCHEMBL9837158 0.67 PYGM (0.46) POLBGAAKDM4EPYGMPYGL
SCHEMBL16178581 0.66 TSHR (0.53) NOTUMGAAKDM4EMEN1KMT2A
SCHEMBL10983420 0.65 MGLL (0.62) MGLLMAPTMEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0234776-B1 PROCESS FOR 1,4-DIHYDROPYRIDINE COMPOUNDS MERCK & CO. INC. (US) 1991-09-04 EP disclosed
US-4780538-A REACTING AN AMINOALKENOATE WITH AN AROMATIC ALDEHYDE USING AN TITANAMINE CATALYST MERCK & CO., INC. (US) 1988-10-25 US disclosed
EP-0234776-A2 Process for 1,4-dihydropyridine compounds MERCK & CO. INC. (US) 1987-09-02 EP disclosed