SCHEMBL9837158

SCHEMBL9837158

C=CCCN1C(C)=C(C(=O)O)C(c2ccccc2)C(C(=O)O)=C1C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PYGM P11217 3/20 0.46
PYGL P06737 2/20 0.46
KDM4E B2RXH2 1/20 0.46
GAA P10253 1/20 0.46
LMNA P02545 4/20 0.42
RECQL P46063 1/20 0.40
APOBEC3A P31941 2/20 0.39
APOBEC3G Q9HC16 2/20 0.39
PABPC1 P11940 1/20 0.38
CACNA1B Q00975 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.36
SIRT3 Q9NTG7 1/20 0.36
POLB P06746 1/20 0.36
TSHR P16473 1/20 0.36
ALDH1A1 P00352 1/20 0.35
CA1 P00915 2/20 0.35
CA2 P00918 2/20 0.35
ADORA3 P0DMS8 1/20 0.35
CACNA1F O60840 1/20 0.34
CACNA1D Q01668 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9836195 0.87 LMNA (0.53) PYGMPYGLKDM4EGAALMNA
SCHEMBL16178523 0.76 KDM4E (0.66) PYGMPYGLKDM4EGAALMNA
SCHEMBL9033367 0.75 PYGM (0.52) PYGMPYGLKDM4EGAALMNA
SCHEMBL11752332 0.74 PYGM (0.49) PYGMPYGLKDM4EGAALMNA
SCHEMBL7328503 0.72 CNR1 (0.44) PYGMPYGLKDM4EGAALMNA
SCHEMBL9833247 0.70 CACNA1B (0.59) PYGMPYGLLMNACACNA1BPOLB
SCHEMBL9836701 0.70 KMT2A (0.49) KDM4EGAALMNARECQLAPOBEC3A
SCHEMBL9033145 0.69 POLB (0.54) PYGMPYGLKDM4EGAALMNA
SCHEMBL9505359 0.69 KDM4E (0.49) PYGMPYGLKDM4EGAALMNA
SCHEMBL11752325 0.69 KDM4E (0.52) PYGMPYGLKDM4EGAALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0234776-B1 PROCESS FOR 1,4-DIHYDROPYRIDINE COMPOUNDS MERCK & CO. INC. (US) 1991-09-04 EP disclosed
US-4780538-A REACTING AN AMINOALKENOATE WITH AN AROMATIC ALDEHYDE USING AN TITANAMINE CATALYST MERCK & CO., INC. (US) 1988-10-25 US disclosed
US-4721708-A CYCLICATION WITH LEWIS ACIDS MERCK & CO., INC. (US) 1988-01-26 US disclosed
EP-0234776-A2 Process for 1,4-dihydropyridine compounds MERCK & CO. INC. (US) 1987-09-02 EP disclosed