SCHEMBL9505457

SCHEMBL9505457

C=CCOC(=O)NCc1ccc(OCC(=O)O)cc1

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 7/20 0.56
EPHX2 P34913 1/20 0.50
NR1H4 Q96RI1 1/20 0.50
FFAR1 O14842 1/20 0.47
KMT2A Q03164 2/20 0.44
HPGD P15428 1/20 0.44
ALOX15 P16050 1/20 0.42
ALDH1A1 P00352 2/20 0.42
MEN1 O00255 1/20 0.42
MAPT P10636 1/20 0.42
PTPN7 P35236 1/20 0.42
PTPN12 Q05209 1/20 0.42
GLA P06280 1/20 0.42
GAA P10253 1/20 0.42
HTT P42858 1/20 0.42
RAB9A P51151 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
ADAMTS5 Q9UNA0 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10418957 0.88 CASP1 (0.49) CASP1FFAR1KMT2AHPGDALDH1A1
SCHEMBL9507749 0.87 CASP1 (0.51) CASP1KMT2AGLA
SCHEMBL14328819 0.82 ALDH1A1 (0.51) CASP1EPHX2NR1H4KMT2AHPGD
SCHEMBL3419896 0.82 CASP1 (0.50) CASP1FFAR1KMT2AALDH1A1MEN1
SCHEMBL7624194 0.81 CASP1 (0.68) CASP1ALDH1A1MAPT
SCHEMBL991422 0.81 CASP1 (0.55) CASP1EPHX2NR1H4FFAR1ALDH1A1
SCHEMBL9508841 0.81 CASP1 (0.52) CASP1KMT2AALOX15ALDH1A1MEN1
SCHEMBL8870036 0.80 CSNK2A2 (0.54) CASP1EPHX2NR1H4FFAR1KMT2A
SCHEMBL992370 0.80 CASP1 (0.53) CASP1KMT2AHPGDALDH1A1MEN1
SCHEMBL991807 0.80 CASP1 (0.53) CASP1EPHX2KMT2AALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0278911-B1 BICYCLIC BETA-LACTAM CARBOXYLIC ACIDS CIBA-GEIGY AG (CH) 1993-08-04 EP disclosed
US-4965260-A PENICILLINS CIBA-GEIGY CORPORATION (US) 1990-10-23 US disclosed
EP-0278911-A1 Bicyclic beta-lactam carboxylic acids CIBA-GEIGY AG (CH) 1988-08-17 EP disclosed