SCHEMBL9508011

SCHEMBL9508011

[CH2]SC1=Nc2ccc(N(C)Cc3ccc(S(=O)(=O)c4ccccc4)cc3)c3cccc1c23

nearest known ligand 0.73

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TYMS P04818 17/20 0.73
HDAC3 O15379 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC11 Q96DB2 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
NCOR2 Q9Y618 1/20 0.38
SCN9A Q15858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9508016 0.89 TYMS (0.58) TYMS
SCHEMBL9080093 0.76 TYMS (1.00) TYMS
SCHEMBL9504568 0.75 TYMS (0.69) TYMS
SCHEMBL9508662 0.72 TYMS (0.59) TYMS
SCHEMBL9506760 0.67 TYMS (0.58) TYMS
Metesind SCHEMBL6703943 0.66 TYMS (1.00) TYMS
SCHEMBL9504724 0.66 TYMS (0.52) TYMS
SCHEMBL9055601 0.66 TYMS (1.00) TYMSHDAC3HDAC1HDAC11HDAC8
SCHEMBL9702076 0.65 TYMS (0.75) TYMS
SCHEMBL9080571 0.65 TYMS (0.79) TYMS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0550566-A1 ANTIPROLIFERATIVE SUBSTITUTED NAPHTHALENE COMPOUNDS AGOURON PHARMACEUTICALS (US) 1993-07-14 EP disclosed
WO-1992005153-A1 ANTIPROLIFERATIVE SUBSTITUTED NAPHTHALENE COMPOUNDS AGOURON PHARMACEUTICALS, INC. (US) 1992-04-02 WO disclosed