SCHEMBL9504568

SCHEMBL9504568

CN(Cc1ccc(S(=O)(=O)c2ccccc2)cc1)C1=Nc2ccc(N)c3cccc1c23

nearest known ligand 0.69

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TYMS P04818 12/20 0.69
HTR6 P50406 1/20 0.36
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
FFAR2 O15552 1/20 0.35
CRHBP P24387 2/20 0.33
CRHR2 Q13324 2/20 0.33
KEAP1 Q14145 1/20 0.33
NFE2L2 Q16236 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9506760 0.88 TYMS (0.58) TYMSHTR6
SCHEMBL9508011 0.75 TYMS (0.73) TYMS
SCHEMBL9508035 0.70 TYMS (0.55) TYMSHTR6FFAR2CRHBPCRHR2
SCHEMBL9508016 0.67 TYMS (0.58) TYMS
SCHEMBL9080093 0.67 TYMS (1.00) TYMSKDM4EALDH1A1
SCHEMBL9704004 0.66 MAPT (0.57) KDM4EALDH1A1KEAP1NFE2L2
SCHEMBL12083406 0.66 ALDH1A1 (0.59) TYMSHTR6ALDH1A1
SCHEMBL9587756 0.65 TYMS (0.43) TYMSHTR6KDM4EALDH1A1CRHBP
SCHEMBL9508662 0.65 TYMS (0.59) TYMSALDH1A1CRHBPCRHR2
SCHEMBL1065778 0.63 DHFR (0.59) TYMS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0550566-A1 ANTIPROLIFERATIVE SUBSTITUTED NAPHTHALENE COMPOUNDS AGOURON PHARMACEUTICALS (US) 1993-07-14 EP disclosed
WO-1992005153-A1 ANTIPROLIFERATIVE SUBSTITUTED NAPHTHALENE COMPOUNDS AGOURON PHARMACEUTICALS, INC. (US) 1992-04-02 WO disclosed