SCHEMBL9508026

SCHEMBL9508026

CCNC1CCCCNC1=O

nearest known ligand 0.58

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.58
CCR2 P41597 18/20 0.55
CCR1 P32246 1/20 0.48
CCR5 P51681 1/20 0.48
CXCR4 P61073 1/20 0.48
RAB9A P51151 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8365578 1.00 HTT (0.58) HTTCCR2CCR1CCR5CXCR4
SCHEMBL13766430 0.94 HTT (0.51) HTTCCR2CCR1CCR5CXCR4
SCHEMBL23374710 0.94 HTT (0.51) HTTCCR2CCR1CCR5CXCR4
SCHEMBL17152685 0.86
SCHEMBL17152686 0.86
SCHEMBL17152684 0.86
SCHEMBL10916213 0.86 CCR2 (0.57) HTTCCR2CCR1CCR5CXCR4
SCHEMBL7098870 0.83 CCR2 (0.58) HTTCCR2CCR1CCR5CXCR4
SCHEMBL8358035 0.82 CCR2 (0.53) HTTCCR2RAB9A
SCHEMBL3008085 0.82 CCR2 (0.53) HTTCCR2RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0294062-B1 RESIN COMPOSITIONS AND MOLDED PRODUCTS THEREOF UBE INDUSTRIES, LTD. (JP) 1993-09-01 EP claimed
US-4879341-A WATERPROOF, FLEXIBILE, RIDIGITY, UBE INDUSTRIES, LTD. (JP) 1989-11-07 US claimed
EP-1813616-B1 Pyrazoloquinolines with immunomodulating activity ACTIVE BIOTECH AB (SE) 2013-03-27 EP disclosed
US-7557110-B2 MAPKAP-K2; inflammatory disease, autoimmune disease, destructive bone disorder, cancer and/or tumour growth; 5-[(trans-4-aminocyclohexyl)amino]-3-fluoro-6-methyl(pyrazolo[1,5-a]pyri- midin-7-yl)}(4-iodophenyl)amine TEIJIN PHARMA LIMITED (JP) 2009-07-07 US disclosed
US-7354946-B2 prominent growth inhibitory activity against tumor cells; cyclin dependent kinase inhibitors; colon cancer; N'-(3-t-butylisoindolino[3,2-b]oxazolidin-4-on-8-yl)-N-(4-(N-benzylpyrrolidin-3-yl)pyridin-2-yl)urea BANYU PHARMACEUTICAL CO., LTD. (JP) 2008-04-08 US disclosed
US-7354946-B2 prominent growth inhibitory activity against tumor cells; cyclin dependent kinase inhibitors; colon cancer; N'-(3-t-butylisoindolino[3,2-b]oxazolidin-4-on-8-yl)-N-(4-(N-benzylpyrrolidin-3-yl)pyridin-2-yl)urea BANYU PHARMACEUTICAL CO., LTD. (JP) 2008-04-08 US disclosed
EP-1562944-B1 PYRAZOLOQUINOLINES WITH IMMUNOMODULATING ACTIVITY ACTIVE BIOTECH AB (SE) 2007-02-14 EP disclosed
US-20070027147-A1 Biarylurea derivatives MSD K.K. (JP) 2007-02-01 US disclosed
US-20070027147-A1 Biarylurea derivatives MSD K.K. (JP) 2007-02-01 US disclosed
EP-0294062-B1 RESIN COMPOSITIONS AND MOLDED PRODUCTS THEREOF UBE INDUSTRIES, LTD. (JP) 1993-09-01 EP disclosed
EP-0128775-B1 RESINOUS COMPOSITION TORAY INDUSTRIES, INC. (JP) 1989-11-15 EP disclosed
US-4879341-A WATERPROOF, FLEXIBILE, RIDIGITY, UBE INDUSTRIES, LTD. (JP) 1989-11-07 US disclosed
EP-0294062-A2 Resin compositions and molded products thereof UBE INDUSTRIES, LTD. (JP) 1988-12-07 EP disclosed
US-4612346-A BLEND OF POLYAMIDE AND MODIFIED POLYOLEFIN TORAY INDUSTRIES, INC. (JP) 1986-09-16 US disclosed
EP-0128775-A2 Resinous composition TORAY INDUSTRIES, INC. (JP) 1984-12-19 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070027147-A1 Biarylurea derivatives CDK6, CDK4, CCNI HTT 3759/4885CCR2 1840/4885CCR1 2580/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.