SCHEMBL9508765

SCHEMBL9508765

Cc1cc(C(=O)CBr)cc(C(=O)O)c1O

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HMGB1 P09429 1/20 0.54
CXCL12 P48061 1/20 0.54
CTH P32929 1/20 0.49
KMT2A Q03164 5/20 0.43
GSK3B P49841 5/20 0.43
MEN1 O00255 3/20 0.43
NPC1 O15118 1/20 0.43
ALDH1A1 P00352 2/20 0.42
KDM4E B2RXH2 1/20 0.42
HPGD P15428 1/20 0.42
HSD17B10 Q99714 1/20 0.42
PTPN1 P18031 4/20 0.41
PHLPP2 Q6ZVD8 1/20 0.39
MAPT P10636 1/20 0.39
AKR1C4 P17516 1/20 0.38
AKR1C3 P42330 1/20 0.38
AKR1C2 P52895 1/20 0.38
AKR1C1 Q04828 1/20 0.38
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9862861 0.85 GSK3B (0.52) KMT2AGSK3BMEN1NPC1ALDH1A1
SCHEMBL4318330 0.84 PTPN1 (0.45) HMGB1CXCL12GSK3BALDH1A1HPGD
SCHEMBL11620046 0.81 HMGB1 (0.53) HMGB1CXCL12CTHKMT2AMEN1
SCHEMBL16056966 0.79 GSK3B (0.55) GSK3BALDH1A1PTPN1
SCHEMBL13645730 0.79 GSK3B (0.46) KMT2AGSK3BMEN1NPC1ALDH1A1
SCHEMBL454210 0.78 HMGB1 (0.56) HMGB1CXCL12CTHKMT2AALDH1A1
SCHEMBL10420496 0.78 HMGB1 (0.53) HMGB1CXCL12CTHKMT2AMEN1
SCHEMBL334660 0.76 HSD17B3 (0.50) HMGB1CXCL12CTHKMT2AMEN1
SCHEMBL9385176 0.75 HMGB1 (0.46) HMGB1CXCL12CTHKMT2AMEN1
SCHEMBL11956604 0.75 GSK3B (0.54) KMT2AGSK3BMEN1NPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0322164-B1 ETHANOLAMINE DERIVATIVES GLAXO GROUP LIMITED (GB) 1993-09-22 EP disclosed
US-5039697-A Adrenergic stimulants, bronchodilators GLAXO GROUP LIMITED (GB) 1991-08-13 US disclosed
US-5032609-A Ethanolamine derivatives GLAXO GROUP LIMITED (GB) 1991-07-16 US disclosed
US-5002966-A Adrenergic Stimulants GLAXO GROUP LIMITED (GB) 1991-03-26 US disclosed
EP-0322164-A2 Ethanolamine derivatives GLAXO GROUP LIMITED (GB) 1989-06-28 EP disclosed