SCHEMBL9510172

SCHEMBL9510172

CCCCCCOc1ccc(C#Cc2ccc(C)cc2)c(F)c1F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.40
HPGD P15428 3/20 0.40
KCNH2 Q12809 1/20 0.39
MAPT P10636 2/20 0.37
THRB P10828 2/20 0.37
NPSR1 Q6W5P4 2/20 0.37
GAA P10253 1/20 0.37
CHUK O15111 1/20 0.35
DAPK3 O43293 1/20 0.35
JAK2 O60674 1/20 0.35
ROCK2 O75116 1/20 0.35
PRKCG P05129 1/20 0.35
CDK1 P06493 1/20 0.35
PIM1 P11309 1/20 0.35
RPS6KB1 P23443 1/20 0.35
CDK2 P24941 1/20 0.35
AKT1 P31749 1/20 0.35
AKT2 P31751 1/20 0.35
MAPKAPK2 P49137 1/20 0.35
BLK P51451 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9511393 0.99 ALDH1A1 (0.38) ALDH1A1HPGDKCNH2MAPTTHRB
SCHEMBL9509499 0.96 ALDH1A1 (0.36) ALDH1A1HPGDKCNH2MAPTTHRB
SCHEMBL9512360 0.95 DRD2 (0.35) ALDH1A1HPGDKCNH2MAPTTHRB
SCHEMBL9509953 0.92 CYP2D6 (0.37) KCNH2L3MBTL1MEN1KMT2A
SCHEMBL9510222 0.91 ACACB (0.35) ALDH1A1KCNH2MAPTGAAKDM4E
SCHEMBL10514590 0.91 MAPT (0.37) ALDH1A1HPGDKCNH2MAPTTHRB
SCHEMBL9508805 0.88 ALDH1A1 (0.39) ALDH1A1HPGDTHRBCHUKDAPK3
SCHEMBL9508826 0.88 AAK1 (0.36) ALDH1A1KCNH2MAPT
SCHEMBL9509482 0.87 HSD17B10 (0.45) ALDH1A1HPGDMAPTTHRBNPSR1
SCHEMBL9512402 0.87 HSD17B10 (0.45) ALDH1A1HPGDMAPTTHRBNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0308438-B1 LIQUID CRYSTAL PHASE CONTAINING TOLANES MERCK PATENT GmbH (DE) 1993-09-29 EP disclosed
EP-0308438-A1 Liquid crystal phase containing tolanes. MERCK PATENT GMBH (DE) 1989-03-29 EP disclosed
WO-1988007514-A1 TOLANES MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1988-10-06 WO disclosed