SCHEMBL9510475

SCHEMBL9510475

COc1ccc(C(O)CCCCCO)c(Cl)c1OC

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 2/20 0.43
TOP1 P11387 4/20 0.40
TUBB1 Q9H4B7 2/20 0.38
ALOX5 P09917 1/20 0.37
SLC2A1 P11166 1/20 0.36
ADRA2A P08913 1/20 0.35
ADRA1A P35348 1/20 0.35
TUBB4A P04350 1/20 0.34
TUBB P07437 1/20 0.34
TUBA3C P0DPH7 1/20 0.34
TUBA1B P68363 1/20 0.34
TUBA4A P68366 1/20 0.34
TUBB4B P68371 1/20 0.34
TUBB3 Q13509 1/20 0.34
TUBB2A Q13885 1/20 0.34
TUBB8 Q3ZCM7 1/20 0.34
TUBA3E Q6PEY2 1/20 0.34
TUBA1A Q71U36 1/20 0.34
TUBA1C Q9BQE3 1/20 0.34
TUBB6 Q9BUF5 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1520565 0.80 ADRA1A (0.54) AOC3TUBB1ADRA2AADRA1ATUBB4A
SCHEMBL22206833 0.76 AOC3 (0.60) AOC3TOP1TUBB1ALOX5ADRA2A
SCHEMBL9509080 0.76 SLC2A1 (0.52) AOC3TUBB1ALOX5SLC2A1TUBB4A
SCHEMBL29234371 0.74 PPARG (0.47) ALOX5ADRA2AADRA1A
SCHEMBL29234372 0.74 PPARG (0.47) ALOX5ADRA2AADRA1A
SCHEMBL9510470 0.72 TUBB1 (0.42) TOP1TUBB1ALOX5TUBB4ATUBB
SCHEMBL10989317 0.72 CYP3A4 (0.45)
SCHEMBL24783647 0.71 TOP1 (0.43) TOP1ALOX5ADRA2AADRA1A
SCHEMBL30859403 0.71 TOP1 (0.43) TOP1ALOX5ADRA2AADRA1A
SCHEMBL29180322 0.71 TOP1 (0.43) TOP1ALOX5ADRA2AADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0310126-B1 DERIVATIVES OF PYROCATECHOL-CARBOXYLIC ACID, THEIR PREPARATION AND USE AS ACTIVE INGREDIENTS IN MEDICINES F. HOFFMANN-LA ROCHE AG (CH) 1993-08-18 EP disclosed
US-5191108-A Lipoxygenase inhibitors, antiinflammatory agents HOFFMANN-LA ROCHE INC. (US) 1993-03-02 US disclosed
US-5025036-A Antiinflammatory agents, gastrointestinal, cardiovascular and skin disorders HOFFMANN-LA ROCHE INC. (US) 1991-06-18 US disclosed
US-4937373-A Substituted naphthalene carboxylic acids HOFFMANN-LA ROCHE INC. (US) 1990-06-26 US disclosed
EP-0310126-A2 Derivatives of pyrocatechol-carboxylic acid, their preparation and use as active ingredients in medicines F. HOFFMANN-LA ROCHE AG (CH) 1989-04-05 EP disclosed