SCHEMBL9510595

SCHEMBL9510595

CC(C)(C)N(NC(=O)c1ccccc1Br)C(=O)c1ccccn1

nearest known ligand 0.64

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 3/20 0.45
POLB P06746 1/20 0.45
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8172818 0.90 ABCB1 (0.47) ABCB1
SCHEMBL9815851 0.87 ABCB1 (0.43) ABCB1POLB
SCHEMBL9815860 0.85 ABCB1 (0.45) ABCB1POLB
SCHEMBL10719304 0.84 ABCB1 (0.56) ABCB1POLB
SCHEMBL9815886 0.83 CTNNB1 (0.52) ABCB1POLB
SCHEMBL8173237 0.82 POLB (0.68) POLB
SCHEMBL9815835 0.81 ABCB1 (0.52) ABCB1
SCHEMBL9510944 0.81 KDM4E (0.49) ABCB1KDM4EALDH1A1
SCHEMBL9714356 0.80 POLB (0.70) ABCB1POLB
SCHEMBL9815854 0.79 ABCB1 (0.58) ABCB1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0361645-B1 ORGANIC HYDRAZINE DERIVATIVES FOR PHARMACEUTICAL USE ROHM AND HAAS COMPANY (US) 1993-09-29 EP disclosed
EP-0253468-B1 SIX-MEMBERED HETEROCYCLIC DERIVATIVES OF N'SUBSTITUTED-N,N'-DIACYLHYDRAZINES ROHM AND HAAS COMPANY (US) 1991-11-06 EP disclosed
EP-0361645-A2 Organic hydrazine derivatives for pharmaceutical use ROHM AND HAAS COMPANY (US) 1990-04-04 EP disclosed