SCHEMBL9510944

SCHEMBL9510944

CC(C)(C)N(NC(=O)c1ccccc1[N+](=O)[O-])C(=O)c1ccccn1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.49
NPC1 O15118 2/20 0.47
RAB9A P51151 2/20 0.47
ALDH1A1 P00352 2/20 0.47
HPGD P15428 1/20 0.46
GAA P10253 1/20 0.45
HTT P42858 1/20 0.45
NCOA1 Q15788 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
NCOA3 Q9Y6Q9 1/20 0.45
ABCB1 P08183 1/20 0.45
CTSD P07339 1/20 0.45
MAPK1 P28482 1/20 0.43
TP53 P04637 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
MAPT P10636 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8173265 0.91 ABCB1 (0.50) KDM4ENPC1RAB9AALDH1A1GAA
SCHEMBL9714633 0.85 ALDH1A1 (0.56) KDM4EALDH1A1ABCB1CTSDMAPT
SCHEMBL9714635 0.82 POLB (0.63) ALDH1A1ABCB1CTSDCYP3A4CYP2C9
SCHEMBL9815860 0.81 ABCB1 (0.45) ABCB1
SCHEMBL9510595 0.81 ABCB1 (0.45) KDM4EALDH1A1ABCB1
SCHEMBL9815833 0.79 ABCB1 (0.66) KDM4ENPC1RAB9AALDH1A1HPGD
SCHEMBL9714479 0.79 ABCB1 (0.55) KDM4ENPC1RAB9AALDH1A1HPGD
SCHEMBL9815886 0.79 CTNNB1 (0.52) GAAABCB1
SCHEMBL8173237 0.78 POLB (0.68) CYP3A4CYP2C9
SCHEMBL10719126 0.78 ABCB1 (0.50) NPC1RAB9AALDH1A1ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0361645-B1 ORGANIC HYDRAZINE DERIVATIVES FOR PHARMACEUTICAL USE ROHM AND HAAS COMPANY (US) 1993-09-29 EP disclosed
EP-0253468-B1 SIX-MEMBERED HETEROCYCLIC DERIVATIVES OF N'SUBSTITUTED-N,N'-DIACYLHYDRAZINES ROHM AND HAAS COMPANY (US) 1991-11-06 EP disclosed
EP-0361645-A2 Organic hydrazine derivatives for pharmaceutical use ROHM AND HAAS COMPANY (US) 1990-04-04 EP disclosed