SCHEMBL9512031

SCHEMBL9512031

CCCc1cc(O)cc(Cl)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 4/20 0.52
CYP3A4 P08684 1/20 0.52
CNR2 P34972 2/20 0.41
CNR1 P21554 1/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
POLB P06746 1/20 0.41
GAA P10253 1/20 0.41
CTDSP1 Q9GZU7 1/20 0.41
LTA4H P09960 1/20 0.40
PTPN1 P18031 1/20 0.40
PTPN11 Q06124 1/20 0.40
GPR84 Q9NQS5 2/20 0.39
HCAR1 Q9BXC0 1/20 0.38
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
MAPT P10636 1/20 0.36
CASP3 P42574 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
SENP8 Q96LD8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26077232 0.84 CNR2 (0.47) PTGS2CYP3A4CNR2CNR1KDM4E
SCHEMBL7634231 0.84 TSHR (0.44) PTGS2CYP3A4CNR2CNR1KDM4E
SCHEMBL28599339 0.84 CNR2 (0.39) PTGS2CYP3A4CNR2CNR1KDM4E
SCHEMBL3362484 0.84 PTGS2 (0.62) PTGS2CYP3A4CNR2CNR1LTA4H
SCHEMBL67909 0.84 PTGS2 (0.70) PTGS2CYP3A4CNR2CNR1LTA4H
SCHEMBL12430083 0.82 CYP3A4 (0.40) PTGS2CYP3A4CNR2CNR1ALDH1A1
SCHEMBL16952302 0.78 CNR2 (0.37) PTGS2CYP3A4CNR2CNR1KDM4E
SCHEMBL16959521 0.78 LTA4H (0.40) PTGS2CYP3A4ALDH1A1LTA4HHCAR1
SCHEMBL2458065 0.78 SMN1; SMN2 (0.38) PTGS2CYP3A4ALDH1A1GPR84HCAR1
SCHEMBL5168458 0.77 PTGS2 (0.56) PTGS2CYP3A4CNR2CNR1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0414686-B1 DERIVATIVES OF TRIFLUOROMETHYL-1-TETRALINES, PREPARATION AND APPLICATION THEREOF FOR THE SYNTHESIS OF COMPOUNDS HAVING THERAPEUTIC PROPERTIES LABORATOIRES LUCIEN (FR) 1993-09-22 EP disclosed
EP-0414686-A1 DERIVATIVES OF TRIFLUOROMETHYL-1-TETRALINES, PREPARATION AND APPLICATION THEREOF FOR THE SYNTHESIS OF COMPOUNDS HAVING THERAPEUTIC PROPERTIES. LUCIEN LAB (FR) 1991-03-06 EP disclosed
WO-1989004819-A1 DERIVATIVES OF TRIFLUOROMETHYL-1-TETRALINES, PREPARATION AND APPLICATION THEREOF FOR THE SYNTHESIS OF COMPOUNDS HAVING THERAPEUTIC PROPERTIES LABORATOIRES LUCIEN (FR) 1989-06-01 WO disclosed