SCHEMBL9512403

SCHEMBL9512403

CC(C)(C)OC(=O)C[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCCC1

nearest known ligand 0.53

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 8/20 0.52
CTSL P07711 5/20 0.51
ITGB3 P05106 1/20 0.50
ITGA2B P08514 1/20 0.50
SYK P43405 1/20 0.49
CTSK P43235 5/20 0.49
CTSS P25774 3/20 0.49
KLK7 P49862 1/20 0.48
KLK5 Q9Y337 1/20 0.48
CASP1 P29466 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9512398 1.00 P2RX7 (0.52) P2RX7CTSLITGB3ITGA2BSYK
SCHEMBL26010144 0.99 CTSL (0.52) P2RX7CTSLITGB3ITGA2BSYK
SCHEMBL16510913 0.92 KLK7 (0.57) P2RX7CTSLITGB3ITGA2BKLK7
SCHEMBL23893528 0.91 CTSL (0.57) P2RX7CTSLITGB3ITGA2BKLK7
SCHEMBL22043924 0.91 CTSL (0.57) P2RX7CTSLITGB3ITGA2BKLK7
SCHEMBL1144124 0.90 P2RX7 (0.57) P2RX7SYK
SCHEMBL1144126 0.90 P2RX7 (0.57) P2RX7SYK
SCHEMBL8882218 0.86 KMT2A (0.47) P2RX7CTSLITGB3ITGA2BCTSK
SCHEMBL6793017 0.85 SYK (0.61) P2RX7CTSLITGB3ITGA2BSYK
SCHEMBL25185922 0.85 CASP1 (0.59) CTSLCTSKCTSSCASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0254545-B1 DIAMINE COMPOUNDS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-10-06 EP disclosed
EP-0254545-A2 Diamine compounds IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1988-01-27 EP disclosed