SCHEMBL9513409

SCHEMBL9513409

O=C(O)CC1(F)N=c2ccccc2=N1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.38
KMT2A Q03164 1/20 0.38
AKR1B1 P15121 2/20 0.35
HSD11B1 P28845 5/20 0.35
PTPN1 P18031 1/20 0.33
GSK3B P49841 1/20 0.33
KEAP1 Q14145 1/20 0.33
CYP2C19 P33261 1/20 0.33
FFAR1 O14842 1/20 0.32
ALOX15 P16050 1/20 0.32
NR4A2 P43354 1/20 0.32
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA3 P07451 1/20 0.32
CA4 P22748 1/20 0.32
CA6 P23280 1/20 0.32
CA5A P35218 1/20 0.32
CA7 P43166 1/20 0.32
CA9 Q16790 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9469517 0.76 PKM (0.38) PKMKMT2AAKR1B1HSD11B1KEAP1
SCHEMBL7352190 0.73 PKM (0.36) PKMKMT2AAKR1B1HSD11B1KEAP1
SCHEMBL17784279 0.67 NPSR1 (0.37) KMT2ACYP2C19ALOX15CA12CA1
SCHEMBL1847048 0.66 PKM (0.37) PKMKMT2AAKR1B1HSD11B1CYP2C19
SCHEMBL8074486 0.66 PKM (0.37) PKMKMT2AAKR1B1HSD11B1TSHR
SCHEMBL7270073 0.66 PKM (0.37) PKMKMT2AAKR1B1HSD11B1TSHR
SCHEMBL9510565 0.65 HTT (0.31) HTT
SCHEMBL15136482 0.64 MAPT (0.36) KMT2ACYP2C19ALOX15CA12CA1
SCHEMBL9112829 0.64 CA12 (0.36) KMT2AGSK3BALOX15CA12CA1
SCHEMBL28956318 0.63 AKR1C1 (0.41) PKMKMT2AALOX15CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0254545-B1 DIAMINE COMPOUNDS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-10-06 EP disclosed
EP-0254545-A2 Diamine compounds IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1988-01-27 EP disclosed