SCHEMBL9514248

SCHEMBL9514248

N#Cc1ccnc(-c2cccc(F)c2)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CLK4 Q9HAZ1 4/20 0.46
ADORA2B P29275 2/20 0.43
ADORA1 P30542 2/20 0.43
ADORA2A P29274 1/20 0.43
KDM4E B2RXH2 1/20 0.43
HPGD P15428 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
RXFP1 Q9HBX9 1/20 0.43
KMO O15229 1/20 0.41
CYP1A2 P05177 2/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2D6 P10635 2/20 0.41
CYP2C19 P33261 2/20 0.41
ALDH1A1 P00352 1/20 0.41
ALOX15 P16050 1/20 0.41
MAPK1 P28482 1/20 0.41
HSD17B10 Q99714 1/20 0.41
LMNA P02545 1/20 0.40
FGFR3 P22607 1/20 0.40
KDR P35968 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6131064 0.80 ABCG2 (0.53) CLK4ADORA1ADORA2AKDM4EHPGD
SCHEMBL27854208 0.76 KMO (0.44) ADORA1ADORA2AKDM4EKMOCYP3A4
SCHEMBL25649075 0.76 NPC1 (0.46) ADORA1ADORA2AKMOGRM5TP53
SCHEMBL4398415 0.75 CLK4 (0.52) CLK4KMOCYP3A4GRM5MAP4K4
SCHEMBL28198548 0.74 CYP2A6 (0.56) CLK4KDM4EHPGDRXFP1CYP1A2
SCHEMBL30629328 0.73 ABCG2 (0.49) RXFP1LMNAGABRG2GABRB3GABRA5
SCHEMBL28547944 0.72 KMO (0.63) ADORA2AKDM4EKMOGRM5MAP4K4
SCHEMBL14153105 0.72 GABRG2 (0.48) ADORA2BADORA1ADORA2AKDM4EHPGD
SCHEMBL27095783 0.71 TAAR1 (0.56) KDM4ETP53
SCHEMBL5739331 0.71 KMO (0.50) ADORA2AKDM4EKMOGRM5MAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0390329-B1 Pyrimidine derivative SEIKO EPSON CORP (JP) 1993-12-01 EP disclosed