SCHEMBL951450

SCHEMBL951450

NC(=O)C(Cc1ccccc1)Cc1cncs1

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.45
SLC6A3 Q01959 1/20 0.43
GPR142 Q7Z601 7/20 0.43
EPHX1 P07099 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
CYP3A4 P08684 4/20 0.42
RAB9A P51151 1/20 0.41
SLC1A3 P43003 1/20 0.41
SLC1A2 P43004 1/20 0.41
SLC1A1 P43005 1/20 0.41
PARP15 Q460N3 1/20 0.41
PARP10 Q53GL7 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5052372 0.79 CYP1A2 (0.68) CYP1A2EPHX1SLC1A3SLC1A2SLC1A1
SCHEMBL3659943 0.73 PARP15 (0.44) SLC6A3TDP1RAB9APARP15PARP10
SCHEMBL9480 0.72 PARP15 (0.43) SLC6A3TDP1RAB9APARP15PARP10
SCHEMBL14637351 0.72 CYP1A2 (0.57) CYP1A2EPHX1SLC1A3SLC1A2SLC1A1
SCHEMBL7437765 0.71 GPR142 (0.51) CYP1A2SLC6A3GPR142EPHX1SLC1A3
SCHEMBL7444446 0.71 CSNK1E (0.44) SLC6A3GPR142EPHX1TDP1CYP3A4
SCHEMBL7179401 0.71 CSNK1E (0.44) SLC6A3GPR142EPHX1TDP1CYP3A4
SCHEMBL19532713 0.71 CYP1A2 (0.61) CYP1A2EPHX1SLC1A3SLC1A2SLC1A1
SCHEMBL7353741 0.71 CYP1A2 (0.61) CYP1A2EPHX1SLC1A3SLC1A2SLC1A1
SCHEMBL6609906 0.71 CYP1A2 (0.61) CYP1A2EPHX1SLC1A3SLC1A2SLC1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2454243-A2 TETRAZOLE DERIVATIVES Merck Serono SA (CH) 2012-05-23 EP disclosed
WO-2011006935-A2 TETRAZOLE DERIVATIVES MERCK SERONO S.A. (CH) 2011-01-20 WO disclosed