SCHEMBL9516044

SCHEMBL9516044

O=P(O)(O)C=CCn1cnc2cncnc21

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FDPS P14324 3/20 0.59
HDAC1 Q13547 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
LTA4H P09960 1/20 0.40
AHCY P23526 5/20 0.35
ALDH1A1 P00352 3/20 0.32
CYP1A2 P05177 3/20 0.32
CYP3A4 P08684 3/20 0.32
CYP2C19 P33261 3/20 0.32
LMNA P02545 2/20 0.32
TSHR P16473 2/20 0.32
CYP2C9 P11712 2/20 0.32
MEN1 O00255 1/20 0.32
HBB P68871 1/20 0.32
KMT2A Q03164 1/20 0.32
USP2 O75604 2/20 0.31
DNMT3B Q9UBC3 1/20 0.31
GGPS1 O95749 1/20 0.31
MAPK1 P28482 1/20 0.30
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4592188 0.81 FDPS (0.51) FDPSHDAC1HDAC6LTA4HAHCY
SCHEMBL4558644 0.77 FDPS (0.54) FDPSHDAC1HDAC6LTA4HAHCY
SCHEMBL3976006 0.74 FDPS (1.00) FDPSHDAC1HDAC6LTA4HALDH1A1
SCHEMBL1079073 0.74 FDPS (0.50) FDPSHDAC1HDAC6LTA4HALDH1A1
SCHEMBL28615898 0.74 AHCY (0.55) FDPSHDAC1HDAC6LTA4HAHCY
SCHEMBL3044440 0.72 FDPS (0.63) FDPSHDAC1HDAC6LTA4HCYP3A4
SCHEMBL8956114 0.71 FDPS (0.56) FDPSHDAC1HDAC6LTA4HALDH1A1
SCHEMBL3054581 0.70 FGFR1 (0.60) FDPSHDAC1HDAC6LTA4HALDH1A1
SCHEMBL1692456 0.70 FDPS (0.56) FDPSHDAC1HDAC6LTA4HALDH1A1
SCHEMBL8708627 0.69 FDPS (0.59) FDPSHDAC1HDAC6LTA4HCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0338887-B1 Phosphonoalkylpurine derivatives MERRELL DOW PHARMA (US) 1993-12-08 EP disclosed
US-4988680-A Phosphorylase inhibitors, immuno suppressants, parasiticides, antileukemia agents MERRELL DOW PHARMACEUTICALS INC. (US) 1991-01-29 US disclosed
EP-0338887-A1 Phosphonoalkylpurine derivatives MERRELL DOW PHARMACEUTICALS INC. (US) 1989-10-25 EP disclosed