SCHEMBL9517705

SCHEMBL9517705

CC(C)C(C)NC(=O)C=CC=C[C@]1(C)C[C@H]1c1ccc(Cl)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.36
HDAC4 P56524 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC7 Q8WUI4 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC10 Q969S8 1/20 0.36
HDAC11 Q96DB2 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
HDAC9 Q9UKV0 1/20 0.36
HDAC5 Q9UQL6 1/20 0.36
NOS3 P29474 2/20 0.34
NOS1 P29475 2/20 0.34
NOS2 P35228 2/20 0.34
P2RX7 Q99572 1/20 0.34
CCR1 P32246 7/20 0.33
MAPK1 P28482 1/20 0.32
MDM2 Q00987 2/20 0.32
TP53 P04637 1/20 0.32
KCNH2 Q12809 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9580474 1.00 HDAC3 (0.36) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL9517708 1.00 HDAC3 (0.36) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL10436499 0.75 CCR2 (0.37) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL9515725 0.75 NOS2 (0.36) NOS3NOS1NOS2
SCHEMBL9519053 0.74 NOS2 (0.34) NOS3NOS1NOS2
SCHEMBL9517700 0.74 KDM1A (0.34) P2RX7MAPK1MDM2TP53LIG1
SCHEMBL9516768 0.70
SCHEMBL9580450 0.68 NOS2 (0.34) NOS3NOS1NOS2LMNAHTT
SCHEMBL9516906 0.68 NOS2 (0.34) NOS3NOS1NOS2LMNAHTT
SCHEMBL9580434 0.68 NOS2 (0.34) NOS3NOS1NOS2LMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0369762-B1 Pesticides ROUSSEL UCLAF (FR) 1993-12-29 EP disclosed
US-5202356-A Insecticides, miticides THE WELLCOME FOUNDATION LIMITED (GB) 1993-04-13 US disclosed
EP-0369762-A1 Pesticides ROUSSEL-UCLAF (FR) 1990-05-23 EP disclosed