SCHEMBL9518535

SCHEMBL9518535

Cc1c(/C=C/C=O)c(-c2ccc(F)cc2)cn1C(C)C

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 8/20 0.54
ADORA2A P29274 1/20 0.33
ADORA1 P30542 1/20 0.33
ABCB1 P08183 1/20 0.33
MET P08581 1/20 0.32
MAPK13 O15264 1/20 0.32
MAPK12 P53778 1/20 0.32
MAPK11 Q15759 1/20 0.32
MAPK14 Q16539 1/20 0.32
PTGS2 P35354 4/20 0.31
PTGDR2 Q9Y5Y4 2/20 0.31
CYP2C9 P11712 1/20 0.30
PTGDR Q13258 1/20 0.30
CDC25A P30304 1/20 0.30
CDC25C P30307 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9750926 1.00 HMGCR (0.54) HMGCRADORA2AADORA1ABCB1MET
SCHEMBL9750845 0.86 HMGCR (0.56) HMGCRADORA2AADORA1ABCB1MET
SCHEMBL9750945 0.85 HMGCR (0.56) HMGCRADORA2AADORA1METMAPK13
SCHEMBL9518437 0.85 HMGCR (0.56) HMGCRADORA2AADORA1METMAPK13
SCHEMBL10397745 0.80 HMGCR (0.38) HMGCRADORA2AADORA1METMAPK13
SCHEMBL10397744 0.80 HMGCR (0.38) HMGCRADORA2AADORA1METMAPK13
SCHEMBL9751002 0.76 HMGCR (0.56) HMGCRABCB1PTGS2
SCHEMBL9751007 0.76 HMGCR (0.56) HMGCRABCB1PTGS2
SCHEMBL31517828 0.75 HMGCR (0.36) HMGCRADORA2AADORA1PTGDR2
SCHEMBL31517692 0.74 HMGCR (0.36) HMGCRMETMAPK13MAPK12MAPK11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0300657-B1 4-SUBSTITUTED 3-OXOBUTANOATE ESTER DERIVATIVES MERCK & CO. INC. (US) 1993-03-31 EP disclosed
EP-0300249-B1 7-[1H-pyrrol-3-yl]-substituted 3,5-dihydroxy-heptane acids, their corresponding delta-lactones and salts, processes for their manufacture, their use as medicines, pharmaceutical preparations and intermediates HOECHST AKTIENGESELLSCHAFT (DE) 1993-02-03 EP disclosed
US-5055484-A Anticholesterol and antilipemic agent HOECHST AKTIENGESELLSCHAFT (DE) 1991-10-08 US disclosed