SCHEMBL9520003

SCHEMBL9520003

COc1cccc(C(=O)c2cccc(F)c2)c1

nearest known ligand 0.74

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 4/20 0.74
NPC1 O15118 3/20 0.74
ALDH1A1 P00352 3/20 0.68
CES2 O00748 2/20 0.62
CES1 P23141 2/20 0.62
STS P08842 3/20 0.60
KDM4E B2RXH2 2/20 0.59
PARP1 P09874 1/20 0.59
SMN1; SMN2 Q16637 2/20 0.57
TSHR P16473 1/20 0.56
NPSR1 Q6W5P4 1/20 0.56
VNN1 O95497 1/20 0.55
POLB P06746 1/20 0.53
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17041600 0.92 RAB9A (0.63) RAB9ANPC1ALDH1A1CES2CES1
SCHEMBL31414638 0.89 CES2 (0.77) RAB9ANPC1CES2CES1STS
SCHEMBL4823687 0.89 CES2 (0.77) RAB9ANPC1CES2CES1STS
SCHEMBL31286476 0.88 STS (0.62) RAB9ANPC1ALDH1A1CES2CES1
SCHEMBL2784166 0.88 ALDH1A1 (0.70) RAB9ANPC1ALDH1A1CES2CES1
Hydrochloric Acid SCHEMBL27733557 0.87 CES2 (0.74) RAB9ANPC1CES2CES1STS
SCHEMBL30414806 0.84 MEN1 (0.69) RAB9ANPC1ALDH1A1CES2CES1
SCHEMBL755443 0.84 MEN1 (0.69) RAB9ANPC1ALDH1A1CES2CES1
SCHEMBL4820908 0.84 CES2 (0.69) RAB9ANPC1CES2CES1STS
SCHEMBL1258944 0.83 CES2 (0.74) RAB9ANPC1CES2CES1PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0299379-B1 PENTADIENAMIDE PAF-ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 1993-04-21 EP disclosed
US-4975438-A ANTICOAGULANT HOFFMANN-LA ROCHE INC. (US) 1990-12-04 US disclosed
EP-0299379-A1 Pentadienamide PAF-antagonists F. HOFFMANN-LA ROCHE AG (CH) 1989-01-18 EP disclosed
US-4788206-A CARDIOVASCULAR DISORDERS, PLATELETS HOFFMANN-LA ROCHE INC. (US) 1988-11-29 US disclosed