SCHEMBL9520601

SCHEMBL9520601

Cc1ccc(NC(=O)N2CC3CC(CN(Cc4ccccc4)C3)C2)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FAAH O00519 6/20 0.62
GRIN2B Q13224 2/20 0.58
CA12 O43570 3/20 0.54
CA2 P00918 3/20 0.54
CA9 Q16790 3/20 0.54
KDM4E B2RXH2 2/20 0.53
MAPT P10636 2/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
MAPK1 P28482 1/20 0.52
NAMPT P43490 1/20 0.51
TAS1R3 Q7RTX0 1/20 0.51
TAS1R1 Q7RTX1 1/20 0.51
TAS1R2 Q8TE23 1/20 0.51
CA1 P00915 2/20 0.49
ALDH1A1 P00352 1/20 0.49
POLB P06746 1/20 0.49
NPC1 O15118 1/20 0.49
TP53 P04637 1/20 0.49
TSHR P16473 1/20 0.49
RAB9A P51151 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6737613 0.91 FAAH (0.66) FAAHGRIN2BCA12CA2CA9
SCHEMBL9520911 0.89 MAPT (0.63) FAAHCA12CA2CA9KDM4E
SCHEMBL9520617 0.88 FAAH (0.55) FAAHGRIN2BCA12CA2CA9
SCHEMBL9519747 0.87 FAAH (0.65) FAAHGRIN2BCA12CA2CA9
SCHEMBL9520201 0.84 FAAH (0.69) FAAHKDM4EMAPTSMN1; SMN2NPC1
SCHEMBL9521948 0.82 ALDH1A1 (0.50) KDM4ESMN1; SMN2MAPK1ALDH1A1POLB
SCHEMBL6732909 0.81 KDM4E (0.50) FAAHKDM4EMAPTSMN1; SMN2ALDH1A1
SCHEMBL6733582 0.80 CYP3A4 (0.46) FAAHKDM4EMAPTSMN1; SMN2ALDH1A1
SCHEMBL10410350 0.79 GAA (0.54) FAAHKDM4EMAPTSMN1; SMN2ALDH1A1
SCHEMBL1895069 0.79 CYP2D6 (0.54) SMN1; SMN2ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0308843-B1 Bispidin derivatives as class III antiarrhythmics BASF AG (DE) 1993-12-15 EP disclosed
US-4959373-A Bispidine derivatives as class III antiarrhythmic agents BASF AKTIENGESELLSCHAFT (DE) 1990-09-25 US disclosed
EP-0308843-A2 Bispidin derivatives as class III antiarrhythmics BASF Aktiengesellschaft (DE) 1989-03-29 EP disclosed