SCHEMBL9520765

SCHEMBL9520765

CCC/C(=C\C=C\CC(=O)O)c1ccc(OC)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 1/20 0.44
PTAFR P25105 1/20 0.43
CA1 P00915 2/20 0.42
CA2 P00918 2/20 0.42
HDAC3 O15379 1/20 0.42
HDAC4 P56524 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC7 Q8WUI4 1/20 0.42
HDAC2 Q92769 1/20 0.42
HDAC10 Q969S8 1/20 0.42
HDAC11 Q96DB2 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
HDAC9 Q9UKV0 1/20 0.42
HDAC5 Q9UQL6 1/20 0.42
TAS1R3 Q7RTX0 1/20 0.42
TAS1R1 Q7RTX1 1/20 0.42
PARP1 P09874 1/20 0.41
PARP10 Q53GL7 1/20 0.41
PARP2 Q9UGN5 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9520959 0.92 PDE4B (0.46) PDE4BPTAFRCA1CA2HDAC3
SCHEMBL9519700 0.91 PTAFR (0.46) PDE4BPTAFRCA1CA2HDAC3
SCHEMBL9519510 0.91 PTAFR (0.46) PDE4BPTAFRCA1CA2HDAC3
SCHEMBL9521062 0.90 PTAFR (0.47) PDE4BPTAFRHDAC3HDAC1HDAC2
SCHEMBL9519702 0.90 PTAFR (0.47) PDE4BPTAFRHDAC3HDAC1HDAC2
SCHEMBL9520661 0.90 PTAFR (0.47) PDE4BPTAFRHDAC3HDAC1HDAC2
SCHEMBL9520013 0.89 CA1 (0.45) PDE4BPTAFRCA1CA2HDAC3
SCHEMBL10398818 0.83 PTAFR (0.49) PDE4BPTAFRCA1CA2HDAC3
Bicarbonate SCHEMBL9520770 0.83 CA1 (0.45) PDE4BPTAFRCA1CA2HDAC3
SCHEMBL10398815 0.83 PTAFR (0.49) PDE4BPTAFRCA1CA2HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0299379-B1 PENTADIENAMIDE PAF-ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 1993-04-21 EP disclosed
EP-0299379-A1 Pentadienamide PAF-antagonists F. HOFFMANN-LA ROCHE AG (CH) 1989-01-18 EP disclosed