SCHEMBL9521134

SCHEMBL9521134

COc1ccc(/C(=C/C=C/CC(=O)O)c2ccccc2OC)cc1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAOB P27338 1/20 0.45
NPC1 O15118 5/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
LMNA P02545 2/20 0.43
CES2 O00748 1/20 0.42
CES1 P23141 1/20 0.42
KMT2A Q03164 3/20 0.42
KCNH2 Q12809 1/20 0.42
MAPT P10636 2/20 0.41
ALDH1A1 P00352 1/20 0.41
GPR52 Q9Y2T5 2/20 0.41
STS P08842 1/20 0.41
RAB9A P51151 3/20 0.40
MEN1 O00255 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
GAA P10253 1/20 0.40
CTSD P07339 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9521080 1.00 MAOB (0.45) MAOBNPC1SMN1; SMN2LMNACES2
SCHEMBL9518925 0.88 GPR52 (0.47) NPC1SMN1; SMN2LMNAKMT2AALDH1A1
SCHEMBL9523136 0.87 CES2 (0.53) MAOBNPC1CES2CES1KMT2A
SCHEMBL9522407 0.87 CES2 (0.53) MAOBNPC1CES2CES1KMT2A
SCHEMBL9521346 0.86 CA1 (0.49) NPC1SMN1; SMN2CES2CES1MAPT
SCHEMBL10398891 0.84 MAOB (0.51) MAOBNPC1SMN1; SMN2LMNACES2
SCHEMBL10399176 0.84 MAOB (0.51) MAOBNPC1SMN1; SMN2LMNACES2
SCHEMBL10398890 0.84 MAOB (0.51) MAOBNPC1SMN1; SMN2LMNACES2
Bicarbonate SCHEMBL9521138 0.84 MAOB (0.48) MAOBNPC1SMN1; SMN2LMNACES2
Bicarbonate SCHEMBL9521090 0.84 MAOB (0.48) MAOBNPC1SMN1; SMN2LMNACES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0299379-B1 PENTADIENAMIDE PAF-ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 1993-04-21 EP disclosed
EP-0299379-A1 Pentadienamide PAF-antagonists F. HOFFMANN-LA ROCHE AG (CH) 1989-01-18 EP disclosed