SCHEMBL9522256

SCHEMBL9522256

c1ccc2cc(CCCN3CCNCC3)ccc2c1

nearest known ligand 0.83

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 3/20 0.83
SIGMAR1 Q99720 11/20 0.67
SLC6A2 P23975 1/20 0.61
SLC6A3 Q01959 1/20 0.61
KCNH2 Q12809 1/20 0.61
HRH3 Q9Y5N1 1/20 0.60
MC4R P32245 1/20 0.49
PKM P14618 1/20 0.49
HTR3E A5X5Y0 1/20 0.47
HTR3B O95264 1/20 0.47
HTR3A P46098 1/20 0.47
HTR5A P47898 1/20 0.47
HTR3D Q70Z44 1/20 0.47
HTR3C Q8WXA8 1/20 0.47
KMT2A Q03164 1/20 0.46
LTA4H P09960 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8671948 0.91 SLC6A4 (1.00) SLC6A4SIGMAR1SLC6A2SLC6A3KCNH2
Hydrochloric Acid SCHEMBL17444691 0.89 SLC6A4 (0.97) SLC6A4SIGMAR1SLC6A2SLC6A3KCNH2
SCHEMBL5604920 0.82 SLC6A4 (0.64) SLC6A4SIGMAR1SLC6A2SLC6A3KCNH2
SCHEMBL593143 0.81 SLC6A4 (0.71) SLC6A4SIGMAR1HRH3MC4RPKM
SCHEMBL457139 0.80 SIGMAR1 (1.00) SIGMAR1LTA4H
SCHEMBL10677264 0.80 SIGMAR1 (1.00) SIGMAR1LTA4H
SCHEMBL16830448 0.80 SLC6A4 (0.69) SLC6A4SIGMAR1HRH3MC4RPKM
SCHEMBL9372748 0.79 SIGMAR1 (1.00) SIGMAR1KCNH2HRH3
SCHEMBL20676401 0.79 SIGMAR1 (0.96) SIGMAR1LTA4H
Hydrochloric Acid SCHEMBL7554612 0.79 SIGMAR1 (0.96) SIGMAR1LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0507863-A4 SIGMA RECEPTOR LIGANDS AND THE USE THEREOF 1993-07-07 EP claimed
EP-0507863-A1 SIGMA RECEPTOR LIGANDS AND THE USE THEREOF VIRGINIA COMMONWEALTH UNIVERSITY (US) 1992-10-14 EP claimed
WO-1991009594-A1 SIGMA RECEPTOR LIGANDS AND THE USE THEREOF VIRGINIA COMMONWEALTH UNIVERSITY (US) 1991-07-11 WO claimed