SCHEMBL9522258

SCHEMBL9522258

c1ccc2c(CCCN3CCNCC3)cccc2c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 5/20 0.60
MC4R P32245 4/20 0.58
TAAR1 Q96RJ0 1/20 0.52
SLC6A4 P31645 2/20 0.50
TDP1 Q9NUW8 2/20 0.50
HTR1A P08908 2/20 0.49
HTR3E A5X5Y0 1/20 0.47
HTR3B O95264 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP2D6 P10635 1/20 0.47
NCF1 P14598 1/20 0.47
TSHR P16473 1/20 0.47
NFKB1 P19838 1/20 0.47
HTR1D P28221 1/20 0.47
HTR1B P28222 1/20 0.47
HTR2A P28223 1/20 0.47
HTR7 P34969 1/20 0.47
MTOR P42345 1/20 0.47
HTR3A P46098 1/20 0.47
HTR5A P47898 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6330371 0.94 MC4R (0.62) SIGMAR1MC4RTAAR1
SCHEMBL2378007 0.91 TDP1 (0.55) SIGMAR1MC4RTAAR1SLC6A4TDP1
Hydrochloric Acid SCHEMBL17444674 0.89 TDP1 (0.54) SIGMAR1MC4RTAAR1SLC6A4TDP1
SCHEMBL4160738 0.82 LMNA (0.53) SIGMAR1MC4RTAAR1SLC6A4TDP1
SCHEMBL1020430 0.81 ACHE (0.62) SIGMAR1SLC6A4HTR1AHTR3EHTR3B
SCHEMBL29567963 0.81 ACHE (0.62) SIGMAR1SLC6A4HTR1AHTR3EHTR3B
SCHEMBL16689990 0.81 ACHE (0.62) SIGMAR1SLC6A4HTR1AHTR3EHTR3B
Bromide SCHEMBL9067059 0.80 ACHE (0.60) SIGMAR1SLC6A4HTR1AHTR3EHTR3B
SCHEMBL16830451 0.80 ACHE (0.60) SIGMAR1SLC6A4HTR1AHTR3EHTR3B
SCHEMBL9378687 0.79 DRD3 (0.64) SIGMAR1MC4RSLC6A4HTR1ACYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0507863-A4 SIGMA RECEPTOR LIGANDS AND THE USE THEREOF 1993-07-07 EP claimed
EP-0507863-A1 SIGMA RECEPTOR LIGANDS AND THE USE THEREOF VIRGINIA COMMONWEALTH UNIVERSITY (US) 1992-10-14 EP claimed
WO-1991009594-A1 SIGMA RECEPTOR LIGANDS AND THE USE THEREOF VIRGINIA COMMONWEALTH UNIVERSITY (US) 1991-07-11 WO claimed