SCHEMBL9523707

SCHEMBL9523707

CCCCn1nnc2cc(CO)ccc21

nearest known ligand 0.63

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HCAR3 P49019 7/20 0.63
SLC9A1 P19634 7/20 0.59
PGR P06401 1/20 0.44
GRM2 Q14416 1/20 0.43
MAPT P10636 1/20 0.41
NAMPT P43490 1/20 0.40
PLA2G4A P47712 1/20 0.40
NR1H2 P55055 1/20 0.39
PPARD Q03181 1/20 0.39
PPARA Q07869 1/20 0.39
NR1H3 Q13133 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3434097 0.84 HCAR3 (0.59) HCAR3SLC9A1MAPTNAMPT
SCHEMBL19848522 0.80 SLC9A1 (0.64) HCAR3SLC9A1GRM2MAPTNAMPT
SCHEMBL19848221 0.79 SLC9A1 (0.62) HCAR3SLC9A1GRM2MAPT
SCHEMBL19848730 0.79 SLC9A1 (0.62) HCAR3SLC9A1GRM2MAPT
SCHEMBL1939333 0.78 HCAR3 (0.54) HCAR3SLC9A1MAPT
SCHEMBL6044071 0.77 HCAR3 (1.00) HCAR3SLC9A1PLA2G4A
SCHEMBL9524513 0.77 HCAR3 (0.50) HCAR3SLC9A1
SCHEMBL19911503 0.77 HCAR3 (0.59) HCAR3SLC9A1GRM2MAPT
SCHEMBL9523866 0.75 HCAR3 (0.61) HCAR3SLC9A1GRM2
SCHEMBL19848183 0.75 HCAR3 (0.58) HCAR3SLC9A1GRM2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0293978-B1 (1H-AZOL-1-YLMETHYL)SUBSTITUTED BENZOTRIAZOLE DERIVATIVES JANSSEN PHARMACEUTICA N.V. (BE) 1993-09-15 EP disclosed
US-5039677-A Estrogen inhibitor JANSSEN PHARMACEUTICA N.V. (CA) 1991-08-13 US disclosed
US-4943574-A AROMATASE INHIBITORS, ESTROGEN DISORDERS JANSSEN PHARMACEUTICA N.V. (BE) 1990-07-24 US disclosed
EP-0293978-A2 (1H-azol-1-ylmethyl)substituted benzotriazole derivatives JANSSEN PHARMACEUTICA N.V. (BE) 1988-12-07 EP disclosed