SCHEMBL9523728

SCHEMBL9523728

c1ccc(CC2(c3ccccc3)CNCCO2)cc1

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 12/20 0.40
SLC6A4 P31645 12/20 0.40
SLC6A3 Q01959 8/20 0.40
HTR2A P28223 1/20 0.40
CYP2D6 P10635 6/20 0.37
KCNH2 Q12809 3/20 0.36
TACR1 P25103 1/20 0.35
OPRM1 P35372 1/20 0.34
MAOA P21397 1/20 0.34
MAOB P27338 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21835471 0.86 CYP3A4 (0.44) SLC6A2SLC6A4SLC6A3CYP2D6OPRM1
SCHEMBL11715846 0.82 HTR2A (0.41) SLC6A2SLC6A4SLC6A3HTR2AOPRM1
SCHEMBL7147295 0.79 HTR2A (0.39) SLC6A2SLC6A4SLC6A3HTR2A
SCHEMBL1036893 0.78 HTR2A (0.38) SLC6A2SLC6A4SLC6A3HTR2AOPRM1
SCHEMBL7008386 0.77 OPRM1 (0.38) SLC6A2SLC6A4SLC6A3HTR2ACYP2D6
SCHEMBL27825135 0.77 TSHR (0.39) SLC6A2SLC6A4SLC6A3HTR2AOPRM1
SCHEMBL15271649 0.77 SLC6A2 (0.34) SLC6A2SLC6A4SLC6A3CYP2D6
SCHEMBL1961851 0.75 SLC6A2 (0.41) SLC6A2SLC6A4SLC6A3HTR2ACYP2D6
SCHEMBL6494298 0.75 MAOA (0.43) OPRM1MAOAMAOB
SCHEMBL6494304 0.75 MAOA (0.43) OPRM1MAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0507863-A4 SIGMA RECEPTOR LIGANDS AND THE USE THEREOF 1993-07-07 EP claimed
EP-0507863-A1 SIGMA RECEPTOR LIGANDS AND THE USE THEREOF VIRGINIA COMMONWEALTH UNIVERSITY (US) 1992-10-14 EP claimed
WO-1991009594-A1 SIGMA RECEPTOR LIGANDS AND THE USE THEREOF VIRGINIA COMMONWEALTH UNIVERSITY (US) 1991-07-11 WO claimed