SCHEMBL9523802

SCHEMBL9523802

COC(=O)c1ccc2c(c1)C(c1cccc[n+]1[O-])=CC(C)(C)O2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARA P10276 2/20 0.40
RARB P10826 2/20 0.40
RARG P13631 2/20 0.40
ALOX5 P09917 1/20 0.40
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
PKM P14618 1/20 0.39
HPGD P15428 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
ABCC9 O60706 2/20 0.39
ABCC8 Q09428 2/20 0.39
KCNJ11 Q14654 2/20 0.39
KCNJ8 Q15842 2/20 0.39
OPRD1 P41143 1/20 0.37
OPRK1 P41145 1/20 0.37
KCNH2 Q12809 1/20 0.37
ABL1 P00519 1/20 0.37
RIN1 Q13671 1/20 0.37
PDK2 Q15119 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9527906 0.88 ABCC9 (0.40) RARARARBRARGKDM4EALDH1A1
SCHEMBL12365140 0.81 RARA (0.55) RARARARBRARGALOX5KDM4E
SCHEMBL9477112 0.80 ALOX5 (0.39) ALOX5KDM4EALDH1A1LMNAPKM
SCHEMBL9525790 0.79 ABCC9 (0.41) RARARARBRARGKDM4EABCC9
SCHEMBL12365911 0.79 RARA (0.43) RARARARBRARGALOX5KDM4E
SCHEMBL9527732 0.78 ABCC9 (0.41) RARARARBRARGABCC9ABCC8
SCHEMBL2263334 0.78 RARA (0.43) RARARARBRARGALOX5KDM4E
SCHEMBL12365916 0.78 NPC1 (0.44) RARARARBRARGALOX5KDM4E
SCHEMBL8335425 0.78 ABCC9 (0.43) ABCC9ABCC8KCNJ11KCNJ8OPRD1
SCHEMBL8796317 0.77 ABCC9 (0.42) ABCC9ABCC8KCNJ11KCNJ8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0298452-B1 2H-1-BENZOPYRANE DERIVATIVES SUBSTITUTED IN POSITION 4 BY ARYL OR N-HETEROARYL F. HOFFMANN-LA ROCHE AG (CH) 1993-06-30 EP claimed
US-5118694-A Hypotensive agents; treatment for cardiovascular and muscular disorders HOFFMANN-LA ROCHE INC. (US) 1992-06-02 US disclosed
US-4971982-A HYPOTENSIVE AGENTS, CARDIOVASCULAR DISORDERS, SMOOTH MUSCLE DISORDERS HOFFMANN-LA ROCHE INC. (US) 1990-11-20 US disclosed