SCHEMBL9524306

SCHEMBL9524306

CC1=C(C(=O)O)C(c2ccccc2C=CC#N)C(C(=O)O)=C(C)N1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.47
CYP3A4 P08684 2/20 0.47
ADORA3 P0DMS8 2/20 0.47
CYP2C9 P11712 2/20 0.47
TBXAS1 P24557 2/20 0.47
CYP2C19 P33261 2/20 0.47
KCNH2 Q12809 2/20 0.47
HTT P42858 2/20 0.47
NR1I2 O75469 2/20 0.47
PGR P06401 1/20 0.47
SLC6A2 P23975 1/20 0.47
DRD3 P35462 1/20 0.47
OPRK1 P41145 1/20 0.47
PDE4D Q08499 1/20 0.47
CACNA1B Q00975 13/20 0.41
KDM4E B2RXH2 3/20 0.39
MAPT P10636 2/20 0.36
ABCC4 O15439 1/20 0.36
PLIN1 O60240 1/20 0.36
CACNA1F O60840 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9524576 1.00 LMNA (0.47) LMNACYP3A4ADORA3CYP2C9TBXAS1
SCHEMBL9524300 1.00 LMNA (0.47) LMNACYP3A4ADORA3CYP2C9TBXAS1
SCHEMBL8595272 0.82 HTT (0.53) LMNACYP3A4ADORA3CYP2C9TBXAS1
SCHEMBL8595275 0.82 HTT (0.53) LMNACYP3A4ADORA3CYP2C9TBXAS1
SCHEMBL9523862 0.81 LMNA (0.39) LMNACYP3A4ADORA3CYP2C9TBXAS1
SCHEMBL9523870 0.81 LMNA (0.39) LMNACYP3A4ADORA3CYP2C9TBXAS1
SCHEMBL9871535 0.81 ADORA3 (0.57) LMNACYP3A4ADORA3CYP2C9TBXAS1
SCHEMBL9871528 0.81 ADORA3 (0.57) LMNACYP3A4ADORA3CYP2C9TBXAS1
SCHEMBL9523854 0.81 LMNA (0.39) LMNACYP3A4ADORA3CYP2C9TBXAS1
SCHEMBL9681769 0.80 LMNA (0.44) LMNACYP3A4ADORA3CYP2C9TBXAS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0245918-B1 1,4-DIHYDROPYRIDINE DERIVATIVES GLAXO S.p.A. (IT) 1993-05-05 EP disclosed
US-4946851-A 1.4-dihydropyridines GLAXO, S.P.A. (IT) 1990-08-07 US disclosed
EP-0245918-A1 1,4-Dihydropyridine derivatives GLAXO S.p.A. (IT) 1987-11-19 EP disclosed