SCHEMBL9525219

SCHEMBL9525219

NC(c1ccccc1)c1c[nH]nn1

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 2/20 0.38
F2 P00734 1/20 0.38
AKT2 P31751 2/20 0.33
SCN4A P35499 2/20 0.32
ADRA2A P08913 1/20 0.31
ADRA2C P18825 1/20 0.31
LMNA P02545 1/20 0.31
HIF1A Q16665 1/20 0.31
CYP19A1 P11511 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5865738 0.80 SLC6A2 (0.45) DPP4F2CYP19A1
SCHEMBL7921340 0.78 CYP19A1 (0.32) DPP4F2AKT2CYP19A1
SCHEMBL1281771 0.77 SMN1; SMN2 (0.40) LMNA
SCHEMBL11351479 0.77 TSHR (0.38) CYP19A1
SCHEMBL15437001 0.77 HTR2C (0.42) ADRA2AADRA2CLMNAHIF1ACYP19A1
SCHEMBL11344228 0.77 CES2 (0.32) CYP19A1
Water SCHEMBL1982282 0.76 SMN1; SMN2 (0.39) LMNA
SCHEMBL2686848 0.74 HTR2A (0.31)
SCHEMBL9634376 0.74 L3MBTL1 (0.35) AKT2
SCHEMBL10560913 0.73 CYP2D6 (0.31) LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105384734-B Trinitrogenazole alcohol antifungal compound and the preparation method and application thereof with the side chain of oxadiazoles containing piperidines 中国人民解放军第二军医大学 2018-07-17 CN disclosed
CN-105384734-A Triazole alcohol antifungal compound with piperidine oxadiazole side chain and preparation method for compound and application of compound UNIV PLA 2ND MILITARY MEDICAL 2016-03-09 CN disclosed
CN-104356125-A Triazole alcohol antifungal compound with side chain containing piperidine oxadiazole as well as preparation method and application thereof UNIV PLA 2ND MILITARY MEDICAL 2015-02-18 CN disclosed
CN-102311399-A Triazole alcohol antifungal compounds with nitrogen-containing side chains, preparation method thereof and application thereof UNIV PLA 2ND MILITARY MEDICAL 2012-01-11 CN disclosed
CN-1303073-C Substituted triazolone benzyl amine triazole antifungal compounds and method for preparing same UNIV PLA 2ND MILITARY MEDICAL (CN) 2007-03-07 CN disclosed
CN-1303073-C Substituted triazolone benzyl amine triazole antifungal compounds and method for preparing same UNIV PLA 2ND MILITARY MEDICAL (CN) 2007-03-07 CN disclosed
CN-1699351-A Substituted triazolone benzyl amine triazole antifungal compounds and method for preparing same UNIV PLA 2ND MILITARY MEDICAL (CN) 2005-11-23 CN disclosed
CN-1699351-A Substituted triazolone benzyl amine triazole antifungal compounds and method for preparing same UNIV PLA 2ND MILITARY MEDICAL (CN) 2005-11-23 CN disclosed
CN-1699351-A Substituted triazolone benzyl amine triazole antifungal compounds and method for preparing same UNIV PLA 2ND MILITARY MEDICAL (CN) 2005-11-23 CN disclosed
EP-0515546-A4 TRIAZOLE ANGIOTENSIN II ANTAGONISTS INCORPORATING A SUBSTITUTED BENZYL ELEMENT 1993-05-12 EP disclosed
EP-0515546-A1 TRIAZOLE ANGIOTENSIN II ANTAGONISTS INCORPORATING A SUBSTITUTED BENZYL ELEMENT MERCK & CO. INC. (US) 1992-12-02 EP disclosed