SCHEMBL9525237

SCHEMBL9525237

COc1cc(NCCO)cc(OC)c1OC

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.47
MAPT P10636 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.44
PTGS2 P35354 1/20 0.44
TUBB4A P04350 2/20 0.44
TUBB P07437 2/20 0.44
TUBA3C P0DPH7 2/20 0.44
TUBA1B P68363 2/20 0.44
TUBA4A P68366 2/20 0.44
TUBB4B P68371 2/20 0.44
TUBB3 Q13509 2/20 0.44
TUBB2A Q13885 2/20 0.44
TUBB8 Q3ZCM7 2/20 0.44
TUBA3E Q6PEY2 2/20 0.44
TUBA1A Q71U36 2/20 0.44
TUBA1C Q9BQE3 2/20 0.44
TUBB6 Q9BUF5 2/20 0.44
TUBB2B Q9BVA1 2/20 0.44
TUBB1 Q9H4B7 2/20 0.44
MEN1 O00255 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23011878 0.84 MAPT (0.50) CYP3A4MAPTSMN1; SMN2PTGS2TUBB4A
SCHEMBL12963092 0.82 PTGS2 (0.50) CYP3A4MAPTSMN1; SMN2PTGS2TUBB4A
SCHEMBL4587193 0.81 PTGS2 (0.44) CYP3A4MAPTSMN1; SMN2PTGS2TUBB4A
SCHEMBL28801415 0.81 HTR2A (0.53) CYP3A4MAPTPTGS2TUBB4ATUBB
SCHEMBL8348474 0.79 KDM4E (0.51) MAPTSMN1; SMN2MEN1KMT2ACYP2C9
SCHEMBL18243936 0.79 MEN1 (0.39) CYP3A4MAPTSMN1; SMN2TUBB4ATUBB
SCHEMBL3207404 0.79 POLB (0.54) CYP3A4MAPTSMN1; SMN2MEN1KMT2A
SCHEMBL2759516 0.78 PTGS2 (0.54) CYP3A4MAPTSMN1; SMN2PTGS2TUBB4A
SCHEMBL13590550 0.77 MAPT (0.47) CYP3A4MAPTSMN1; SMN2PTGS2TUBB4A
SCHEMBL5162466 0.77 POLB (0.44) SMN1; SMN2TUBB4ATUBBTUBA3CTUBA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0301751-B1 PYRIDINIUM DERIVATIVES, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1993-03-10 EP disclosed
US-4962113-A PLATELET ACTIVATING FACTOR ANTAGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD (JP) 1990-10-09 US disclosed
EP-0301751-A1 Pyridinium derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1989-02-01 EP disclosed