SCHEMBL9525255

SCHEMBL9525255

O=C(NCCOc1cccc2ccccc12)OCCN(C(=O)c1cncc(Cl)c1)c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.44
ALDH1A1 P00352 3/20 0.44
HPGD P15428 2/20 0.44
HRH4 Q9H3N8 1/20 0.39
HRH3 Q9Y5N1 1/20 0.39
MCL1 Q07820 3/20 0.37
BCL2 P10415 2/20 0.37
BCL2L1 Q07817 2/20 0.37
KMT2A Q03164 2/20 0.37
HTR1B P28222 3/20 0.36
HTR1D P28221 2/20 0.36
ATM Q13315 1/20 0.36
TRPM4 Q8TD43 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
POLB P06746 1/20 0.35
G6PD P11413 1/20 0.35
MCHR1 Q99705 1/20 0.35
BAD Q92934 1/20 0.35
SLC6A4 P31645 1/20 0.35
HRH1 P35367 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9524147 0.90 KDM4E (0.44) KDM4EALDH1A1HPGDHRH4HRH3
SCHEMBL9524584 0.87 KDM4E (0.41) KDM4EALDH1A1HPGDHRH4HRH3
Iodide SCHEMBL9523929 0.82 KDM4E (0.41) KDM4EALDH1A1HPGDMCL1KMT2A
Hydrochloric Acid SCHEMBL9525954 0.82 KDM4E (0.41) KDM4EALDH1A1HPGDMCL1KMT2A
SCHEMBL9525095 0.80 CFTR (0.42) KDM4EALDH1A1HPGDKMT2AHTR1B
SCHEMBL10401410 0.79 LMNA (0.47) KDM4EALDH1A1HPGDKMT2ASMN1; SMN2
SCHEMBL9525232 0.78 KDM4E (0.44) KDM4EALDH1A1HPGDMCL1KMT2A
SCHEMBL9523896 0.77 KDM4E (0.43) KDM4EALDH1A1HPGDKMT2AHTR1B
SCHEMBL9524400 0.76 ALDH1A1 (0.41) KDM4EALDH1A1HPGDSMN1; SMN2POLB
Iodide SCHEMBL9528125 0.76 KDM4E (0.42) KDM4EALDH1A1HPGDKMT2AHTR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0301751-B1 PYRIDINIUM DERIVATIVES, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1993-03-10 EP disclosed
US-4962113-A PLATELET ACTIVATING FACTOR ANTAGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD (JP) 1990-10-09 US disclosed
EP-0301751-A1 Pyridinium derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1989-02-01 EP disclosed