SCHEMBL9525418

SCHEMBL9525418

O=C=Nc1ccc(-c2ccc(C(F)(F)F)cc2)s1

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PRF1 P14222 1/20 0.39
KIF11 P52732 8/20 0.36
WRN Q14191 1/20 0.36
MKNK1 Q9BUB5 1/20 0.34
MKNK2 Q9HBH9 1/20 0.34
HDAC6 Q9UBN7 3/20 0.33
HDAC1 Q13547 2/20 0.33
HDAC4 P56524 1/20 0.33
BACE1 P56817 1/20 0.33
HSD17B2 P37059 1/20 0.32
JAK2 O60674 1/20 0.32
STK17B O94768 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9524424 0.84 NPC1 (0.38) KIF11WRNHDAC6HDAC1
SCHEMBL3045728 0.78 RAB9A (0.42) HDAC6HDAC1HSD17B2
SCHEMBL27961778 0.76 KIF11 (0.52) PRF1KIF11HSD17B2
SCHEMBL14705447 0.76 KIF11 (0.52) PRF1KIF11HSD17B2
SCHEMBL14705469 0.74 KIF11 (0.50) PRF1KIF11WRNMKNK1MKNK2
SCHEMBL25165734 0.73 KIF11 (0.54) PRF1KIF11HSD17B2
SCHEMBL27274253 0.72 DAO (0.41)
SCHEMBL332062 0.70 CYP3A4 (0.37)
SCHEMBL28473667 0.70 KIF11 (0.68) KIF11HDAC6BACE1HSD17B2
SCHEMBL160983 0.69 CYP3A4 (0.50) KIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0259972-B1 HETEROCYCLIC PROPENE AMIDE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS PHARMACEUTICALS LILLY INDUSTRIES LIMITED (GB) 1993-07-14 EP disclosed
US-4983619-A Leukotriene antagonists LILLY INDUSTRIES LIMITED (GB) 1991-01-08 US disclosed
EP-0259972-A2 Heterocyclic propene amide derivatives, processes for their preparation and their use as pharmaceuticals LILLY INDUSTRIES LIMITED (GB) 1988-03-16 EP disclosed