SCHEMBL9525569

SCHEMBL9525569

CCCCc1noc(NS(=O)(=O)c2ccc(F)cc2)c1Cc1ccc(-c2ccccc2)c(-c2nnn[nH]2)c1

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 1/20 0.38
FFAR4 Q5NUL3 1/20 0.38
EDNRA P25101 5/20 0.36
METAP2 P50579 1/20 0.35
EDNRB P24530 4/20 0.35
TRPV1 Q8NER1 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9526834 0.92 FFAR1 (0.39) FFAR1FFAR4EDNRAEDNRB
SCHEMBL9526402 0.82 ADRB2 (0.39) EDNRAEDNRB
SCHEMBL9525332 0.82 AGTR2 (0.38) METAP2
SCHEMBL9526466 0.79
SCHEMBL9527525 0.79 AGTR1 (0.38)
SCHEMBL9525968 0.78 FFAR1 (0.39) FFAR1FFAR4
SCHEMBL9527711 0.77 PPARG (0.33)
SCHEMBL9529965 0.76 AGTR1 (0.40)
SCHEMBL9527727 0.75 AGTR2 (0.41)
SCHEMBL9530326 0.74

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0523141-A4 SUBSTITUTED PYRAZOLES, ISOXAZOLES AND ISOTHIAZOLES 1993-04-21 EP disclosed
EP-0523141-A1 SUBSTITUTED PYRAZOLES, ISOXAZOLES AND ISOTHIAZOLES MERCK & CO. INC. (US) 1993-01-20 EP disclosed