SCHEMBL9525860

SCHEMBL9525860

CC(C)(C)OC(=O)c1ccc2c(c1)-c1c(c(C(=O)Cl)nn1-c1ccccc1)CS2

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TP53 P04637 4/20 0.38
PIK3CD O00329 6/20 0.37
PIK3R2 O00459 6/20 0.37
PIK3CA P42336 6/20 0.37
PIK3CB P42338 6/20 0.37
PIK3CG P48736 6/20 0.37
PIK3R5 Q8WYR1 6/20 0.37
PIK3R3 Q92569 6/20 0.37
MAPT P10636 5/20 0.37
LMNA P02545 2/20 0.37
ALDH1A1 P00352 2/20 0.35
CYP3A4 P08684 2/20 0.35
CYP2C9 P11712 2/20 0.35
CYP2C19 P33261 2/20 0.35
NPSR1 Q6W5P4 1/20 0.35
PTGS1 P23219 1/20 0.35
PTGS2 P35354 1/20 0.35
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9522810 0.93 TP53 (0.39) TP53PIK3CDPIK3R2PIK3CAPIK3CB
SCHEMBL9523046 0.88 ALDH1A1 (0.46) TP53MAPTALDH1A1CYP3A4CYP2C9
SCHEMBL9827669 0.85 PTGS1 (0.35) TP53PIK3CDPIK3R2PIK3CAPIK3CB
SCHEMBL9526026 0.81 ALDH1A1 (0.48) TP53MAPTALDH1A1CYP3A4CYP2C9
SCHEMBL9522746 0.81 TP53 (0.37) TP53PIK3CDPIK3R2PIK3CAPIK3CB
SCHEMBL9523265 0.80 TP53 (0.53) TP53MAPTPTGS1PTGS2
SCHEMBL9523795 0.77 ALDH1A1 (0.50) TP53MAPTALDH1A1CYP3A4CYP2C9
SCHEMBL9523022 0.74 MAPT (0.42) TP53MAPTLMNA
SCHEMBL12275859 0.72 PIK3CD (0.46) TP53PIK3CDPIK3R2PIK3CAPIK3CB
SCHEMBL12276272 0.72 ALDH1A1 (0.48) TP53MAPTLMNAALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0420883-B1 TRICYCLIC 3-OXO-PROPANENITRILE DERIVATIVES AND PROCESS FOR THEIR PREPARATION ERBA CARLO SPA (IT) 1993-11-03 EP disclosed