SCHEMBL9526328

SCHEMBL9526328

O=C(c1ccccc1)N(CCO)CCCN(C(=O)O)c1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2C P18825 1/20 0.54
LPAR1 Q92633 1/20 0.45
HDAC1 Q13547 4/20 0.43
HDAC6 Q9UBN7 4/20 0.43
HDAC3 O15379 2/20 0.43
HDAC4 P56524 2/20 0.43
HDAC2 Q92769 2/20 0.43
HDAC10 Q969S8 2/20 0.43
HDAC8 Q9BY41 2/20 0.43
NCOR2 Q9Y618 1/20 0.43
KMT2A Q03164 2/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
LIMK2 P53671 1/20 0.42
LTB4R2 Q9NPC1 2/20 0.42
GAA P10253 2/20 0.42
TSHR P16473 1/20 0.42
HDAC7 Q8WUI4 1/20 0.41
HDAC11 Q96DB2 1/20 0.41
HDAC9 Q9UKV0 1/20 0.41
HDAC5 Q9UQL6 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7791465 0.82 HDAC3 (0.51) ADRA2CHDAC1HDAC6HDAC3HDAC4
SCHEMBL154607 0.82 HPGD (0.53) ADRA2CHDAC1HDAC6HDAC3HDAC4
Hydrochloric Acid SCHEMBL27871652 0.81 HPGD (0.52) ADRA2CLPAR1HDAC1HDAC6HDAC3
SCHEMBL7751510 0.79 ADRA2C (0.69) ADRA2CHDAC1HDAC6HDAC3HDAC4
SCHEMBL4918307 0.79 ADRA2C (0.50) ADRA2CHDAC1HDAC6HDAC3HDAC4
SCHEMBL7543305 0.77 HPGD (0.43) ADRA2CLPAR1HDAC1HDAC6HDAC3
SCHEMBL5154776 0.77 ADRA2C (0.55) ADRA2CKMT2AGAATSHRMEN1
SCHEMBL8615545 0.76 LIMK2 (0.63) LPAR1HDAC1HDAC6HDAC3HDAC4
SCHEMBL10925719 0.76 HPGD (0.56) HDAC1HDAC6HDAC3HDAC2LTB4R2
SCHEMBL30957362 0.75 NPC1 (0.57) ADRA2CHDAC1HDAC3HDAC2HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0301751-B1 PYRIDINIUM DERIVATIVES, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1993-03-10 EP disclosed
US-4962113-A PLATELET ACTIVATING FACTOR ANTAGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD (JP) 1990-10-09 US disclosed
EP-0301751-A1 Pyridinium derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1989-02-01 EP disclosed