SCHEMBL9526674

SCHEMBL9526674

O=C(CBr)c1ccc(C(F)(F)F)cc1Cl

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 1/20 0.54
GSK3B P49841 1/20 0.54
CES2 O00748 2/20 0.46
ALDH1A1 P00352 4/20 0.44
KDM4E B2RXH2 1/20 0.44
HPGD P15428 1/20 0.44
HSD17B10 Q99714 1/20 0.44
MRGPRX4 Q96LA9 3/20 0.43
PDE2A O00408 2/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
MAPK1 P28482 1/20 0.42
HIF1A Q16665 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C19 P33261 1/20 0.42
RAB9A P51151 1/20 0.42
SORT1 Q99523 1/20 0.42
AVPR2 P30518 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1198647 0.87 PTPN1 (0.54) PTPN1GSK3BCES2ALDH1A1HPGD
SCHEMBL5951860 0.83 PDE2A (0.50) CES2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL30634441 0.81 PTPN1 (0.56) PTPN1GSK3BCES2ALDH1A1KDM4E
SCHEMBL2097720 0.81 CES2 (0.66) PTPN1GSK3BCES2ALDH1A1KDM4E
SCHEMBL1960700 0.81 PTPN1 (0.56) PTPN1GSK3BCES2ALDH1A1KDM4E
SCHEMBL30006617 0.81 PTPN1 (0.56) PTPN1GSK3BCES2ALDH1A1KDM4E
SCHEMBL7786271 0.81 PTPN1 (0.56) PTPN1GSK3BCES2ALDH1A1KDM4E
SCHEMBL21462078 0.81 PTPN1 (0.56) PTPN1GSK3BCES2ALDH1A1KDM4E
SCHEMBL8617573 0.81 KDM4E (0.61) CES2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL8493470 0.81 ALDH1A1 (0.48) CES2ALDH1A1KDM4EHPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5142092-A Chemical intermediate for making fungicides BAYER AKTIENGESELLSCHAFT (DE) 1992-08-25 US claimed
EP-0365914-B1 FLUORINE-CONTAINING ACETOPHENONES OPTIONALLY HALOGENATED IN THE CH3-GROUP, AND THEIR PREPARATION FROM FLUORINATED BENZONITRILES BAYER AG (DE) 1992-07-22 EP claimed
EP-0365914-A2 Fluorine-containing acetophenones optionally halogenated in the CH3-group, and their preparation from fluorinated benzonitriles BAYER AG (DE) 1990-05-02 EP claimed
EP-0365913-B1 Substituted 2-aminothiazoles BAYER AG (DE) 1993-11-18 EP disclosed
US-5142092-A Chemical intermediate for making fungicides BAYER AKTIENGESELLSCHAFT (DE) 1992-08-25 US disclosed
EP-0365914-B1 FLUORINE-CONTAINING ACETOPHENONES OPTIONALLY HALOGENATED IN THE CH3-GROUP, AND THEIR PREPARATION FROM FLUORINATED BENZONITRILES BAYER AG (DE) 1992-07-22 EP disclosed
US-5104879-A ANTIMYCOTICALLY ACTIVE SUBSTITUTED 2-AMINOTHIAZOLES BAYER AKTIENGESELLSCHAFT (DE) 1992-04-14 US disclosed