SCHEMBL9526953

SCHEMBL9526953

CCCc1nsc(C(=O)O)c1Cc1ccc(-c2ccccc2S(=O)(=O)NC(=O)C(c2ccccc2)c2ccccc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AGTR2 P50052 7/20 0.47
AGTR1 P30556 5/20 0.47
TBXA2R P21731 1/20 0.39
PTGER1 P34995 1/20 0.39
PTGER4 P35408 1/20 0.39
PTGFR P43088 1/20 0.39
PTGER3 P43115 1/20 0.39
PTGIR P43119 1/20 0.39
PTGDR Q13258 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9526081 0.87 AGTR2 (0.53) AGTR2AGTR1
SCHEMBL9525641 0.85 AGTR1 (0.49) AGTR2AGTR1
SCHEMBL9530087 0.83 AGTR2 (0.47) AGTR2AGTR1TBXA2RPTGER1PTGER4
SCHEMBL9527786 0.83 AGTR2 (0.47) AGTR2AGTR1TBXA2RPTGER1PTGER4
SCHEMBL9530400 0.82 AGTR2 (0.57) AGTR2AGTR1
SCHEMBL9527244 0.81 AGTR2 (0.46) AGTR2AGTR1
SCHEMBL9526473 0.81 AGTR1 (0.47) AGTR2AGTR1
SCHEMBL9531915 0.78 AGTR2 (0.46) AGTR2AGTR1
SCHEMBL9526726 0.78 AGTR1 (0.50) AGTR2AGTR1TBXA2RPTGER1PTGER4
SCHEMBL9526539 0.75 AGTR2 (0.41) AGTR2AGTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0523141-A4 SUBSTITUTED PYRAZOLES, ISOXAZOLES AND ISOTHIAZOLES 1993-04-21 EP claimed
EP-0523141-A1 SUBSTITUTED PYRAZOLES, ISOXAZOLES AND ISOTHIAZOLES MERCK & CO. INC. (US) 1993-01-20 EP claimed
WO-1991015479-A1 SUBSTITUTED PYRAZOLES, ISOXAZOLES AND ISOTHIAZOLES MERCK & CO., INC. (US) 1991-10-17 WO claimed